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Found 7 Enz. Inhib. hit(s) with all data for entry = 50044046
TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50366820(BULLATACIN)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
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TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50004703(Corossoline)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
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TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50004702((10S)-COROSSOLINE)
Affinity DataIC50:  2nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
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TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50004705(CIS-SOLAMIN)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
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TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50004705(CIS-SOLAMIN)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
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TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50004701((17R,18R,21R,22S)-reticulation-1)
Affinity DataIC50:  16nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
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TargetNADH-ubiquinone oxidoreductase chain 1(Bos taurus (Bovine))TBA
LigandPNGBDBM50004700((17S, 18S, 21S, 22R)-reticulation-1)
Affinity DataIC50:  17nMAssay Description:Inhibition of Bos taurus (bovine) mitochodrial complex 1 isolated from heart submitochondrial particle by NADH oxidase assayMore data for this Ligand-Target Pair
In DepthDetails Article