Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50044255
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010383BDBM50010383(CHEMBL3263959)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 28031BDBM28031(N-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorop...)
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010382BDBM50010382(CHEMBL3263958)
Affinity DataIC50: 7nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5446BDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50315887BDBM50315887((1s,3s)-3-(8-amino-1-(2-phenylquinolin-7-yl)imidaz...)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010383BDBM50010383(CHEMBL3263959)
Affinity DataIC50: 39nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010386BDBM50010386(CHEMBL3263962)
Affinity DataIC50: 84nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010388BDBM50010388(CHEMBL3263964)
Affinity DataIC50: 94nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010387BDBM50010387(CHEMBL3263963)
Affinity DataIC50: 168nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010382BDBM50010382(CHEMBL3263958)
Affinity DataIC50: 170nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010388BDBM50010388(CHEMBL3263964)
Affinity DataIC50: 398nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010386BDBM50010386(CHEMBL3263962)
Affinity DataIC50: 564nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010389BDBM50010389(CHEMBL3263965)
Affinity DataIC50: 572nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010384BDBM50010384(CHEMBL3263960)
Affinity DataIC50: 978nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010387BDBM50010387(CHEMBL3263963)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010392BDBM50010392(CHEMBL3263968)
Affinity DataIC50: 1.05E+3nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010391BDBM50010391(CHEMBL3263967)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010390BDBM50010390(CHEMBL3263966)
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010385BDBM50010385(CHEMBL3263961)
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010389BDBM50010389(CHEMBL3263965)
Affinity DataIC50: 1.66E+3nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010385BDBM50010385(CHEMBL3263961)
Affinity DataIC50: 1.72E+3nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010393BDBM50010393(CHEMBL3263969)
Affinity DataIC50: 1.91E+3nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010391BDBM50010391(CHEMBL3263967)
Affinity DataIC50: 2.69E+3nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010393BDBM50010393(CHEMBL3263969)
Affinity DataIC50: 2.71E+3nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010392BDBM50010392(CHEMBL3263968)
Affinity DataIC50: 2.71E+3nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010388BDBM50010388(CHEMBL3263964)
Affinity DataIC50: 2.87E+3nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010384BDBM50010384(CHEMBL3263960)
Affinity DataIC50: 3.86E+3nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010390BDBM50010390(CHEMBL3263966)
Affinity DataIC50: 4.35E+3nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010387BDBM50010387(CHEMBL3263963)
Affinity DataIC50: 5.23E+3nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010383BDBM50010383(CHEMBL3263959)
Affinity DataIC50: 7.67E+3nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010386BDBM50010386(CHEMBL3263962)
Affinity DataIC50: 7.87E+3nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010389BDBM50010389(CHEMBL3263965)
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5446BDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetHepatocyte growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50315887BDBM50315887((1s,3s)-3-(8-amino-1-(2-phenylquinolin-7-yl)imidaz...)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant c-MET (unknown origin) using poly-AEKY peptide as substrate after 60 mins by ADPGlo assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010393BDBM50010393(CHEMBL3263969)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 5446BDBM5446(Erlotinib | OSI-774 | N-(3-ethynylphenyl)-6,7-bis(...)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 28031BDBM28031(N-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorop...)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010390BDBM50010390(CHEMBL3263966)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010391BDBM50010391(CHEMBL3263967)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010392BDBM50010392(CHEMBL3263968)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 28031BDBM28031(N-{4-[(2-amino-3-chloropyridin-4-yl)oxy]-3-fluorop...)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010384BDBM50010384(CHEMBL3263960)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50315887BDBM50315887((1s,3s)-3-(8-amino-1-(2-phenylquinolin-7-yl)imidaz...)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetInsulin receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010385BDBM50010385(CHEMBL3263961)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant INSR (unknown origin) using fluorescent dye-labelled KKSRGDYMTMQIG peptide peptide as substrate after 1 hr by IMAP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50306682BDBM50306682((R)-3-(1-(2,6-dichloro-3-fluorophenyl)ethoxy)-5-(1...)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Vichem Chemie Research

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50010382BDBM50010382(CHEMBL3263958)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of recombinant EGFR (unknown origin) using poly-GT peptide as substrate by Transcreener assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2015
Entry Details Article
PubMed