Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 50045441
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062762BDBM50062762(CHEMBL3397792)
Affinity DataKi:  0.710nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062765BDBM50062765(CHEMBL3397793)
Affinity DataKi:  2.70nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062769BDBM50062769(CHEMBL3397803)
Affinity DataKi:  4.80nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062752BDBM50062752(CHEMBL3397805)
Affinity DataKi:  4.90nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062755BDBM50062755(CHEMBL3397798)
Affinity DataKi:  5.90nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062760BDBM50062760(CHEMBL3397809)
Affinity DataKi:  7.40nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062769BDBM50062769(CHEMBL3397803)
Affinity DataKi:  8.90nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062764BDBM50062764(CHEMBL3397800)
Affinity DataKi:  9nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062766BDBM50062766(CHEMBL3397801)
Affinity DataKi:  9.30nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062753BDBM50062753(CHEMBL3397806)
Affinity DataKi:  10nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062761BDBM50062761(CHEMBL3397810)
Affinity DataKi:  13nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062760BDBM50062760(CHEMBL3397809)
Affinity DataKi:  13nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062770BDBM50062770(CHEMBL3397804)
Affinity DataKi:  17nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062759BDBM50062759(CHEMBL3397808)
Affinity DataKi:  20nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062762BDBM50062762(CHEMBL3397792)
Affinity DataKi:  25nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062770BDBM50062770(CHEMBL3397804)
Affinity DataKi:  26nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062752BDBM50062752(CHEMBL3397805)
Affinity DataKi:  26nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062768BDBM50062768(CHEMBL3397802)
Affinity DataKi:  27nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062755BDBM50062755(CHEMBL3397798)
Affinity DataKi:  27nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062759BDBM50062759(CHEMBL3397808)
Affinity DataKi:  28nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062768BDBM50062768(CHEMBL3397802)
Affinity DataKi:  29nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062761BDBM50062761(CHEMBL3397810)
Affinity DataKi:  29nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062763BDBM50062763(CHEMBL3397807)
Affinity DataKi:  29nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062757BDBM50062757(CHEMBL3397795)
Affinity DataKi:  30nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062767BDBM50062767(CHEMBL3397794)
Affinity DataKi:  34nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062765BDBM50062765(CHEMBL3397793)
Affinity DataKi:  34nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062753BDBM50062753(CHEMBL3397806)
Affinity DataKi:  37nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062756BDBM50062756(CHEMBL3397799)
Affinity DataKi:  38nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062756BDBM50062756(CHEMBL3397799)
Affinity DataKi:  42nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062764BDBM50062764(CHEMBL3397800)
Affinity DataKi:  42nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062758BDBM50062758(CHEMBL3397796)
Affinity DataKi:  44nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062756BDBM50062756(CHEMBL3397799)
Affinity DataKi:  44nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062764BDBM50062764(CHEMBL3397800)
Affinity DataKi:  48nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062766BDBM50062766(CHEMBL3397801)
Affinity DataKi:  52nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062770BDBM50062770(CHEMBL3397804)
Affinity DataKi:  54nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062763BDBM50062763(CHEMBL3397807)
Affinity DataKi:  57nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062757BDBM50062757(CHEMBL3397795)
Affinity DataKi:  59nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062766BDBM50062766(CHEMBL3397801)
Affinity DataKi:  64nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062768BDBM50062768(CHEMBL3397802)
Affinity DataKi:  68nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062762BDBM50062762(CHEMBL3397792)
Affinity DataKi:  82nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062769BDBM50062769(CHEMBL3397803)
Affinity DataKi:  107nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062763BDBM50062763(CHEMBL3397807)
Affinity DataKi:  129nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetTransporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062754BDBM50062754(CHEMBL3397797)
Affinity DataKi:  152nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat cerebral cortex NETMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062767BDBM50062767(CHEMBL3397794)
Affinity DataKi:  167nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062758BDBM50062758(CHEMBL3397796)
Affinity DataKi:  209nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062767BDBM50062767(CHEMBL3397794)
Affinity DataKi:  223nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062765BDBM50062765(CHEMBL3397793)
Affinity DataKi:  234nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062759BDBM50062759(CHEMBL3397808)
Affinity DataKi:  258nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent dopamine transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062754BDBM50062754(CHEMBL3397797)
Affinity DataKi:  259nMAssay Description:Inhibition of [ring 2,5,6-3H]dopamine reuptake in rat striatum DATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
TargetSodium-dependent serotonin transporter(Rat)
Wayne State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50062757BDBM50062757(CHEMBL3397795)
Affinity DataKi:  281nMAssay Description:Inhibition of [1,2-3H]serotonin reuptake in rat cerebral cortex SERTMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/7/2016
Entry Details Article
PubMed
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