Affinity DataEC50: 1.61E+3nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 3.23E+3nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 720nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 310nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 410nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 250nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: >3.30E+4nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 3.17E+3nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 460nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 2.69E+3nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 6.34E+3nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 220nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 490nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 2.37E+3nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 2.25E+3nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 6.19E+3nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 7.69E+3nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 670nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 1.52E+4nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 1.03E+3nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 2.21E+4nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 1.83E+3nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 340nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair
Affinity DataEC50: 3.03E+3nMAssay Description:Antagonist activity against S1P1R in human U2OS cells expressing beta-arrestin/green fluorescent protein assessed as effect on S1P-induced beta-arres...More data for this Ligand-Target Pair