Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 50046146
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50422013(Lobeline Hydrochloride | LOBELINE)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]-nicotine from alpha4beta2 nicotine acetylcholine receptor (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50364890(Amixin IC | TILORONE | cid_5475)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]-MLA from alpha7 nicotine acetylcholine receptor in rat brain minus cerebellum after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50088438(CHEMBL71085 | 1-Pyridin-3-yl-[1,4]diazepane | NS35...)
Affinity DataIC50: 190nMAssay Description:Displacement of [3H]-alpha-bungarotoxin from alpha7 nicotine acetylcholine receptor in Wistar rat cerebral cortex after 2 hrs by liquid scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50096271(CHEMBL3593679)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-MLA from Sprague-Dawley rat brain alpha7 nicotine acetylcholine receptor after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50096270(CHEMBL3593678)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-MLA from Sprague-Dawley rat brain alpha7 nicotine acetylcholine receptor after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098558(CHEMBL3593852)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-MLA from Sprague-Dawley rat brain alpha7 nicotine acetylcholine receptor after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098559(CHEMBL3593851)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50096269(CHEMBL3593677)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098558(CHEMBL3593852)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50096270(CHEMBL3593678)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098557(CHEMBL3593853)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50096271(CHEMBL3593679)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50096274(CHEMBL3593844)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50096275(CHEMBL3593845)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098460(CHEMBL3593846)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098445(CHEMBL3593849)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-MLA from Sprague-Dawley rat brain alpha7 nicotine acetylcholine receptor after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098450(CHEMBL3593847)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098449(CHEMBL3593848)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50096273(CHEMBL3593843)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-MLA from Sprague-Dawley rat brain alpha7 nicotine acetylcholine receptor after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098445(CHEMBL3593849)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098444(CHEMBL3593850)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50096272(CHEMBL3593842)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-MLA from Sprague-Dawley rat brain alpha7 nicotine acetylcholine receptor after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50096272(CHEMBL3593842)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50096273(CHEMBL3593843)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098542(CHEMBL3593855)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098469(CHEMBL3593859)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-MLA from Sprague-Dawley rat brain alpha7 nicotine acetylcholine receptor after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098541(CHEMBL3593856)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098539(CHEMBL3593857)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098538(CHEMBL3593858)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Human)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098469(CHEMBL3593859)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity to alpha3beta4 nicotine acetylcholine receptor (unknown origin) after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098542(CHEMBL3593855)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-MLA from Sprague-Dawley rat brain alpha7 nicotine acetylcholine receptor after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098539(CHEMBL3593857)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-MLA from Sprague-Dawley rat brain alpha7 nicotine acetylcholine receptor after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50098541(CHEMBL3593856)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-MLA from Sprague-Dawley rat brain alpha7 nicotine acetylcholine receptor after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50096269(CHEMBL3593677)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]-MLA from Sprague-Dawley rat brain alpha7 nicotine acetylcholine receptor after 90 mins by radioligand displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50096268(CHEMBL3593676)
Affinity DataIC50: 4.60E+3nMAssay Description:Displacement of [3H]-alpha-bungarotoxin from alpha7 nicotine acetylcholine receptor in Wistar rat cerebral cortex after 2 hrs by liquid scintillation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rat)
University of Hawaii At Hilo

Curated by ChEMBL
LigandPNGBDBM50422013(Lobeline Hydrochloride | LOBELINE)
Affinity DataKi:  6.60E+3nMAssay Description:Displacement of [3H]-methyllycaconitine from alpha7 nicotine acetylcholine receptor in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/18/2016
Entry Details Article
PubMed