Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 50048218
TargetAurora kinase A(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50334594(2-(5-chloro-2-(2-methoxy-4-morpholinophenylamino)p...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human AURKAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM192755(TG101209 | US11643396, Example TG101209 | US112797...)
Affinity DataIC50: 6nMAssay Description:Inhibition of human JAK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetTyrosine-protein kinase JAK2(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208589(CHEMBL3884848)
Affinity DataIC50: 50nMAssay Description:Inhibition of human JAK2 using poly (Glu:Tyr) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208590(CHEMBL3884104)
Affinity DataIC50: 126nMAssay Description:Inhibition of human JAK2 using poly (Glu:Tyr) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208588(CHEMBL3884240)
Affinity DataIC50: 129nMAssay Description:Inhibition of human JAK2 using poly (Glu:Tyr) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208592(CHEMBL3883652)
Affinity DataIC50: 140nMAssay Description:Inhibition of human JAK2 using poly (Glu:Tyr) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208589(CHEMBL3884848)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human JAK3 using poly (Glu:Tyr) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208592(CHEMBL3883652)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of human JAK3 using poly (Glu:Tyr) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208590(CHEMBL3884104)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of human JAK3 using poly (Glu:Tyr) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208588(CHEMBL3884240)
Affinity DataIC50: 7.10E+3nMAssay Description:Inhibition of human JAK3 using poly (Glu:Tyr) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208592(CHEMBL3883652)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of human EGFR using poly (Glu:Tyr) as substrate measured for 1.5 hrs by oregon green 488 dye-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208588(CHEMBL3884240)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human EGFR using poly (Glu:Tyr) as substrate measured for 1.5 hrs by oregon green 488 dye-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK3(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208591(CHEMBL3885292)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JAK3 using poly (Glu:Tyr) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetTyrosine-protein kinase JAK2(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208591(CHEMBL3885292)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human JAK2 using poly (Glu:Tyr) as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208590(CHEMBL3884104)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of human EGFR using poly (Glu:Tyr) as substrate measured for 1.5 hrs by oregon green 488 dye-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208589(CHEMBL3884848)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of human EGFR using poly (Glu:Tyr) as substrate measured for 1.5 hrs by oregon green 488 dye-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed
TargetEpidermal growth factor receptor(Human)
Kasetsart University

Curated by ChEMBL
LigandPNGBDBM50208591(CHEMBL3885292)
Affinity DataIC50: 1.50E+5nMAssay Description:Inhibition of human EGFR using poly (Glu:Tyr) as substrate measured for 1.5 hrs by oregon green 488 dye-based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2018
Entry Details Article
PubMed