Compile Data Set for Download or QSAR
maximum 50k data
Found 29 Enz. Inhib. hit(s) with all data for entry = 50048629
LigandPNGBDBM50223718(CHEMBL273788)
Affinity DataIC50:  9nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50452855(Isoptpo Hyoscine | Scopolamine)
Affinity DataIC50:  10nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223771(CHEMBL14668)
Affinity DataIC50:  11nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataIC50:  11nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50017536((Flumezapine)7-Fluoro-2-methyl-10-(4-methyl-pipera...)
Affinity DataIC50:  20nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223714(CHEMBL14995)
Affinity DataIC50:  26nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223662(CHEMBL276753)
Affinity DataIC50:  26nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223713(CHEMBL276095)
Affinity DataIC50:  31nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223663(CHEMBL14766)
Affinity DataIC50:  34nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223659(CHEMBL14427)
Affinity DataIC50:  64nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50017536((Flumezapine)7-Fluoro-2-methyl-10-(4-methyl-pipera...)
Affinity DataIC50:  74nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223659(CHEMBL14427)
Affinity DataIC50:  75nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223663(CHEMBL14766)
Affinity DataIC50:  77nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223712(CHEMBL274043)
Affinity DataIC50:  91nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223711(CHEMBL278473)
Affinity DataIC50:  93nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223713(CHEMBL276095)
Affinity DataIC50:  97nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223660(CHEMBL14605)
Affinity DataIC50:  101nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223771(CHEMBL14668)
Affinity DataIC50:  116nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223714(CHEMBL14995)
Affinity DataIC50:  172nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataIC50:  179nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223662(CHEMBL276753)
Affinity DataIC50:  180nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223661(CHEMBL276754)
Affinity DataIC50:  199nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223718(CHEMBL273788)
Affinity DataIC50:  223nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223711(CHEMBL278473)
Affinity DataIC50:  247nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50001884(2-[4-(4-Methyl-benzyl)-piperazin-1-yl]-1-(2-methyl...)
Affinity DataIC50:  247nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223712(CHEMBL274043)
Affinity DataIC50:  258nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50223661(CHEMBL276754)
Affinity DataIC50:  574nMAssay Description:Displacement of [3H]QNB from Muscarinic acetylcholine receptor of rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50223660(CHEMBL14605)
Affinity DataIC50:  624nMAssay Description:Displacement of [3H]spiroperidol from Dopamine receptor of rat striatum membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataIC50: >1.00E+4nMAssay Description:The ability to displace [3H]QNB from Muscarinic acetylcholine receptor in rat brain membrane was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed