Compile Data Set for Download or QSAR
Report error Found 45 Enz. Inhib. hit(s) with all data for entry = 4804
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM81498(5-Methoxy-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-i...)
Affinity DataKi:  9.77nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50024206(3-[2-(dimethylamino)ethyl]indol-5-ol | 5-hydroxy-N...)
Affinity DataKi:  21.4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  29.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM30704(METERGOLINE | (phenylmethyl) N-[[(6aR,9S,10aR)-4,7...)
Affinity DataKi:  34.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM30707(3-(2-DIMETHYLAMINOETHYL)-5-METHOXYINDOLE | CHEMBL7...)
Affinity DataKi:  39.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM10755([3H]-5-HT | 5-Hydroxy Tryptamine | 2-imino-1-methy...)
Affinity DataKi:  46.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50031942(CHEMBL1065 | Sansert | (6aR,9R)-4-Methyl-4,6,6a,7,...)
Affinity DataKi:  70.8nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM78940(methanesulfonic acid;1-methyl-4-(3-methylsulfanyl-...)
Affinity DataKi:  89.1nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50014945(alpha-methyl-5-HT | alpha-methyl-5-hydroxytryptami...)
Affinity DataKi:  158nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM30704(METERGOLINE | (phenylmethyl) N-[[(6aR,9S,10aR)-4,7...)
Affinity DataKi:  245nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM30707(3-(2-DIMETHYLAMINOETHYL)-5-METHOXYINDOLE | CHEMBL7...)
Affinity DataKi:  288nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM82087(tryptamine, 5-Methoxy | 5-Methoxytryptamine hydroc...)
Affinity DataKi:  288nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50014945(alpha-methyl-5-HT | alpha-methyl-5-hydroxytryptami...)
Affinity DataKi:  501nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50001859(BUSPAR | CHEMBL49 | 8-[4-(4-Pyrimidin-2-yl-piperaz...)
Affinity DataKi:  891nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM81498(5-Methoxy-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-i...)
Affinity DataKi:  912nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50017721(5-(1-methylpiperidylidene-4)-5H-dibenzo(a,d)cyclop...)
Affinity DataKi:  977nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50024206(3-[2-(dimethylamino)ethyl]indol-5-ol | 5-hydroxy-N...)
Affinity DataKi:  1.02E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50016900(CINANSERIN | CHEMBL18786 | N-(2-(3-(dimethylamino)...)
Affinity DataKi:  1.10E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM78940(methanesulfonic acid;1-methyl-4-(3-methylsulfanyl-...)
Affinity DataKi:  1.15E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50014407(2-Piperazin-1-yl-quinoline (Quipazine) | CHEMBL187...)
Affinity DataKi:  1.17E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  1.32E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50013515(yohimbic acid methyl ester | 17alpha-hydroxyyohimb...)
Affinity DataKi:  1.55E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM82088(NSC_27400 | CAS_15574-96-6 | PIZOTIFEN)
Affinity DataKi:  2.19E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50014407(2-Piperazin-1-yl-quinoline (Quipazine) | CHEMBL187...)
Affinity DataKi:  3.39E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  3.55E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50024210(1H-indole-3-ethanamine | CHEMBL6640 | 2-(3-indolyl...)
Affinity DataKi:  3.72E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  4.17E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM21395(3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}e...)
Affinity DataKi:  4.17E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50031942(CHEMBL1065 | Sansert | (6aR,9R)-4-Methyl-4,6,6a,7,...)
Affinity DataKi:  4.68E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50017721(5-(1-methylpiperidylidene-4)-5H-dibenzo(a,d)cyclop...)
Affinity DataKi:  5.25E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM82088(NSC_27400 | CAS_15574-96-6 | PIZOTIFEN)
Affinity DataKi:  6.17E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM35234(Noradrenaline,(+) | NOREPINEPHRINE | DL-[7-3H]nore...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM35234(Noradrenaline,(+) | NOREPINEPHRINE | DL-[7-3H]nore...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM82087(tryptamine, 5-Methoxy | 5-Methoxytryptamine hydroc...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50017696(N,N,alpha-trimethyl-10H-phenothiazine-10-ethanamin...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50017696(N,N,alpha-trimethyl-10H-phenothiazine-10-ethanamin...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM86698(CHEMBL116590 | CAS_132-17-2 | NSC_2344 | BENZTROPI...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM86698(CHEMBL116590 | CAS_132-17-2 | NSC_2344 | BENZTROPI...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50016900(CINANSERIN | CHEMBL18786 | N-(2-(3-(dimethylamino)...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50024210(1H-indole-3-ethanamine | CHEMBL6640 | 2-(3-indolyl...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50010859(CHEMBL11 | Imipramin | IMIPRAMINE HYDROCHLORIDE | ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM55121(cid_65340 | Dopamine | SMR000059081 | 4-(2-aminoet...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM21395(3-(2-{4-[(4-fluorophenyl)carbonyl]piperidin-1-yl}e...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Rat)
College of France

Curated by PDSP Ki Database
LigandPNGBDBM50010859(CHEMBL11 | Imipramin | IMIPRAMINE HYDROCHLORIDE | ...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/27/2011
Entry Details Article
PubMed