Compile Data Set for Download or QSAR
Report error Found 654 Enz. Inhib. hit(s) with all data for entry = 357
TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263706BDBM263706(6-(2- chloro-4- ethoxy- phenyl)-5- [4-[(3S)-1- (3-...)
Affinity DataIC50: 0.800nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263911BDBM263911(US9714221, Example 207)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263755BDBM263755(6-(2- chloro-4- methoxy- phenyl)-5- [4-[(3S)-1- (3...)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263709BDBM263709(6-(4- ethoxy-2- methyl- phenyl)-1- fluoro-5-[4- [(...)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263847BDBM263847(6-(2,2-dimethylindolin-5-yl)-5-[4-[(3S)-1-(3-fluor...)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263748BDBM263748(US9714221, Example 82)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263737BDBM263737(6-(6- ethoxy-2- fluoro-3- pyridyl)-5- [4-[(3S)- 1-...)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263712BDBM263712(6-(2,3- dihydro- 1,4- benzodioxin-6-yl)-5- [4-[(3S...)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263900BDBM263900(6-[2,3- difluoro-4- (1-piperidyl)- phenyl]-5- [4-[...)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263860BDBM263860(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263893BDBM263893(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263892BDBM263892(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263743BDBM263743(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263775BDBM263775(US9714221, Example 109)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263764BDBM263764(6-(2,2- dimethyl- 3H- benzo- furan-5-yl)-5- [4-[(3...)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263707BDBM263707(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263774BDBM263774(US9714221, Example 108)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263719BDBM263719(6-(1,3- benzoxazol- 5-yl)-5-[4- [(3S)-1-(3- fluoro...)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263710BDBM263710(6-(2,4- dichloro- phenyl)-1- fluoro-5-[4- [(3S)-1-...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263692BDBM263692(US9714221, Example 29)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263759BDBM263759(6-(2,3- difluoro-4- methoxy- phenyl)-5- [4-[(3S)-1...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263691BDBM263691(6- (benzofuran- 5-yl)-5- [4-[(3S)-1- (3- fluoropro...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263850BDBM263850(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263669BDBM263669(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263736BDBM263736(US9714221, Example 70)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263801BDBM263801(6-(2,2- difluoro- 1,3- benzo- dioxol-5-yl)-5- [4-[...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263757BDBM263757(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263673BDBM263673(6-(2-fluoro- 4-hydroxy- phenyl)-5- [4-[(3S)-1- (3-...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263740BDBM263740(6-(3-ethoxy- phenyl)-5-[4- [(3S)-1-(3- fluoropropy...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263694BDBM263694(6-(2,3- dimethyl- phenyl)-5-[4- [(3S)-1-(3- fluoro...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263717BDBM263717(6-(4- ethoxy- 2,3- difluoro- phenyl)-5- [4-[(3S)-1...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263782BDBM263782(6-[4- (difluoro- methoxy)-2- fluoro- phenyl]-5- [4...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor [Y537S](Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263692BDBM263692(US9714221, Example 29)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263697BDBM263697(6-(6- ethoxy-3- pyridyl)-5- [4-[(3S)-1- (3- fluoro...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263742BDBM263742(US9714221, Example 76)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263674BDBM263674(US9714221, Example 11)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263806BDBM263806(6-(6- ethoxy-4- methyl-3- pyridyl)-5- [4-[(3S)-1- ...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263907BDBM263907(US9714221, Example 203)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263723BDBM263723(6-(2- chlorophenyl)- 5-[4- [(3S)-1-(3- fluoropropy...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263788BDBM263788(6-(2- chloro-3- fluoro- phenyl)-1- fluoro-5-[4- [(...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263834BDBM263834(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263813BDBM263813(6-[4- (difluoro- methoxy)-2- methyl- phenyl]-5- [4...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263724BDBM263724(2-[5-[4- [(3S)-1-(3- fluoropropyl)- pyrrolidin-3- ...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263917BDBM263917(6-(2-chloro-4-fluoro-phenyl)-1-fluoro-5-[4-[(3S)-1...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263705BDBM263705(6-(4- ethoxy-2- fluoro- phenyl)-5- [4-[(3S)-1- (3-...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263843BDBM263843(6-(6- ethoxy-5- fluoro-3- pyridyl)-5- [4-[(3S)-1- ...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263683BDBM263683(5-[4-[(3S)- 1-(3- fluoropropyl)- pyrrolidin-3- yl]...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263770BDBM263770(6-(2-fluoro- 6-methoxy- 3-pyridyl)- 5-[4-[(3S)- 1-...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263708BDBM263708(US9714221, Example 45)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

TargetEstrogen receptor(Human)
Sanofi

US Patent
LigandChemical structure of BindingDB Monomer ID 263896BDBM263896(6-(2,1,3- benzothia- diazol-5-yl)- 5-[4-[(3S)- 1-(...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:It is a competition assay, where binding of a test compound to a complex comprised of (i) His6-ERα298-554 protein representing ERα ligand-b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2018
Entry Details
US Patent

Displayed 1 to 50 (of 654 total ) | Next | Last >>
Jump to: