Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50040217
TargetSolute carrier family 15 member 2(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50016695((2S)-2-{[(2S)-2-aminopropanoyl]amino}propanoic aci...)
Affinity DataKi:  6.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT2-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSolute carrier family 15 member 2(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50169217(6-Amino-2-(2-amino-3-carboxy-propionylamino)-hexan...)
Affinity DataKi:  8.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT2-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSolute carrier family 15 member 2(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50169125(Ala-Lys | (S)-6-Amino-2-((S)-2-amino-propionylamin...)
Affinity DataKi:  1.10E+4nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT2-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSolute carrier family 15 member 2(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50188504(Ala-Asp | CHEMBL380047)
Affinity DataKi:  1.80E+4nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT2-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSolute carrier family 15 member 2(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50169138((S)-2-((S)-2,6-Diamino-hexanoylamino)-propionic ac...)
Affinity DataKi:  2.30E+4nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT2-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50016695((2S)-2-{[(2S)-2-aminopropanoyl]amino}propanoic aci...)
Affinity DataKi:  7.80E+4nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50188504(Ala-Asp | CHEMBL380047)
Affinity DataKi:  7.80E+4nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50169217(6-Amino-2-(2-amino-3-carboxy-propionylamino)-hexan...)
Affinity DataKi:  1.08E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50169125(Ala-Lys | (S)-6-Amino-2-((S)-2-amino-propionylamin...)
Affinity DataKi:  1.17E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSolute carrier family 15 member 1(Human)
Medical College of Georgia

Curated by ChEMBL
LigandPNGBDBM50169138((S)-2-((S)-2,6-Diamino-hexanoylamino)-propionic ac...)
Affinity DataKi:  4.19E+5nMAssay Description:TP_TRANSPORTER: inhibition of Gly-Sar uptake in PEPT1-expressing HeLa cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed