TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.00E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 7.94nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.58E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.58E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Rattus norvegicus)
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 2.51E+3nMAssay Description:Tested antagonist activity toward NK-3 receptor in rat portal vein against the agonist eledoisinMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.26E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 2.51E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 398nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Tested for antagonist activity toward NK-1 receptor in guinea pig ileum against the agonist eledoisinMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Rattus norvegicus)
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.26E+4nMAssay Description:Tested for antagonist activity toward NK-3 receptor in rat portal vein against the agonist eledoisinMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.00E+3nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.00E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
Affinity DataKd: 2.00E+3nMAssay Description:Tested for antagonist activity toward NK-1 receptor in guinea pig ileum against the agonist eledoisin (mean +/-, n=4)More data for this Ligand-Target Pair
Affinity DataKd: 251nMAssay Description:Tested for antagonist activity toward NK-1 receptor in guinea pig ileum against the agonist eledoisinMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 7.94E+3nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Rattus norvegicus)
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Tested for antagonist activity toward NK-3 receptor in rat portal vein against the agonist eledoisinMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 200nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 2.00E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Rattus norvegicus)
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 3.98E+3nMAssay Description:Tested for antagonist activity toward NK-3 receptor in rat portal vein against the agonist eledoisinMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 1.00E+4nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 631nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetSubstance-K receptor(Rattus norvegicus (Rat))
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 2.51E+3nMAssay Description:Inhibition of eledoisin binding to NK-2 receptor in rat vas deferensMore data for this Ligand-Target Pair
TargetNeuromedin-K receptor(Rattus norvegicus)
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Merck Sharp And Dohme Research Laboratories
Curated by ChEMBL
Affinity DataKd: 7.94E+3nMAssay Description:Tested for antagonist activity toward NK-3 receptor in rat portal vein against the agonist eledoisin (mean +/-, n=4)More data for this Ligand-Target Pair