Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50005194
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034128(CHEMBL441396 | Neuropeptide Y(NPY) | Tyr-Pro-Ser-L...)
Affinity DataIC50:  0.450nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034111(CHEMBL269515 | Tyr-Ile-Asn-Leu-Ile-Tyr-Arg-Leu-Arg...)
Affinity DataIC50:  8nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034118(CHEMBL274850 | His-Tyr-Ile-Asn-Leu-Ile-Tyr-Arg-Leu...)
Affinity DataIC50:  12nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034116(Arg-His-Tyr-Ile-Asn-Leu-Ile-Tyr-Arg-Leu-Arg-Tyr-NH...)
Affinity DataIC50:  12nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034125(CHEMBL265849 | Neuropeptide Y(NPY)(13-36) | Pro-Al...)
Affinity DataIC50:  15nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034127(CHEMBL409457 | Ile-Asn-Leu-Ile-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataIC50:  37nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034113(CHEMBL385246 | Tyr-Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg...)
Affinity DataIC50:  44nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034123(CHEMBL439534 | NPY[Tyr32,Leu34])
Affinity DataIC50:  83nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034121(CHEMBL386823 | Ile-Asn-Pro-Ile-Tyr-Arg-Leu-Arg-Tyr...)
Affinity DataIC50:  174nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034120(Asn-Leu-Ile-Tyr-Arg-Leu-Arg-Tyr-NH2 | CHEMBL428097)
Affinity DataIC50:  310nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034126(CHEMBL439356 | Tyr-Ile-Asn-Leu-Leu-Tyr-Arg-Gln-Arg...)
Affinity DataIC50:  370nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034124(1N-[1-[4-amino(imino)methylamino-1-(1-{4-amino(imi...)
Affinity DataIC50:  400nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034114(Arg-His-Tyr-Ile-Asn-Leu-Ile-Thr-Arg-Gln-Arg-Tyr-NH...)
Affinity DataIC50:  1.30E+3nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034117(CHEMBL406275 | Tyr-Ile-Asn-Leu-Ile-Thr-Arg-Leu-Tyr...)
Affinity DataIC50:  2.10E+3nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034112(CHEMBL269544 | Tyr-Ile-Asn-Leu-Leu-Tyr-Arg-Pro-Arg...)
Affinity DataIC50:  2.70E+3nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034129(1N-[1-[4-amino(imino)methylamino-1-(1-{4-amino(imi...)
Affinity DataIC50:  2.95E+3nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034119(CHEMBL385245 | Tyr-Ile-Asn-Leu-Ile-Thr-Arg-Gln-Arg...)
Affinity DataIC50:  3.00E+4nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034115(1N-[1-carbamoyl-2-phenyl-(1S)-ethyl]-5-amino(imino...)
Affinity DataIC50:  4.00E+4nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y receptor type 2(RAT)
Burroughs Wellcome

Curated by ChEMBL
LigandPNGBDBM50034122(1N-{4-amino(imino)methylamino-1-[1-carbamoyl-2-(4-...)
Affinity DataIC50: >1.00E+5nMAssay Description:50% displacement of specifically bound [3H]-NPY2 from rat brain membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed