Compile Data Set for Download or QSAR
maximum 50k data
Found 170 Enz. Inhib. hit(s) with all data for entry = 50005295
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035320((+/-)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035303((R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035305((S)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035335((R)-8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035326(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035324((S)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM21393(7-(dipropylamino)-5,6,7,8-tetrahydronaphthalen-1-o...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035319(8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  0.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035315((S)-8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035328((R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035304((4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035307(CHEMBL302171 | Dipropyl-(S)-6,7,8,9-tetrahydro-3H-...)
Affinity DataKi:  1.40nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035317(((R)-4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-...)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035304((4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity against Dopamine receptor D3 from CHO-K1 cells, using [3H]-spiperone as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035306((1-Chloro-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  2nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035313(8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035304((4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  2.80nMAssay Description:Binding affinity against Dopamine receptor D2 from CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035329((+/-)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  3.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035299(((S)-4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-...)
Affinity DataKi:  3.70nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035299(((S)-4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-...)
Affinity DataKi:  4.10nMAssay Description:Binding affinity against Dopamine receptor D3 from CHO-K1 cells, using [3H]-spiperone as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035299(((S)-4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity against Dopamine receptor D2 from CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035335((R)-8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H...)
Affinity DataKi:  4.40nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035319(8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  4.60nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035330(CHEMBL302172 | Dipropyl-(R)-6,7,8,9-tetrahydro-3H-...)
Affinity DataKi:  5.20nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035325((4-Fluoro-1-propyl-6,7,8,9-tetrahydro-3H-benzo[e]i...)
Affinity DataKi:  5.90nMAssay Description:Binding affinity against Dopamine receptor D2 from CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035328((R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  6.70nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035300(1-(8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H-...)
Affinity DataKi:  7.10nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035322(2-(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]i...)
Affinity DataKi:  7.30nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035330(CHEMBL302172 | Dipropyl-(R)-6,7,8,9-tetrahydro-3H-...)
Affinity DataKi:  7.40nMAssay Description:Binding affinity against Dopamine receptor D2 expressed in CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035326(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  7.5nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035317(((R)-4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-...)
Affinity DataKi:  7.80nMAssay Description:Binding affinity against Dopamine receptor D2 from CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035325((4-Fluoro-1-propyl-6,7,8,9-tetrahydro-3H-benzo[e]i...)
Affinity DataKi:  8.40nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035313(8-Dipropylamino-4-fluoro-6,7,8,9-tetrahydro-3H-ben...)
Affinity DataKi:  8.60nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035316((8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]ind...)
Affinity DataKi:  8.60nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035306((1-Chloro-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  9.80nMAssay Description:Binding affinity against Dopamine receptor D2 expressed in CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035308(8-Dipropylamino-1,3,6,7,8,9-hexahydro-benzo[e]indo...)
Affinity DataKi:  11nMAssay Description:Binding affinity against Dopamine receptor D2 from CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035325((4-Fluoro-1-propyl-6,7,8,9-tetrahydro-3H-benzo[e]i...)
Affinity DataKi:  11nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035309((1-Methanesulfonyl-6,7,8,9-tetrahydro-3H-benzo[e]i...)
Affinity DataKi:  11nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035304((4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  11nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035310((1-Methyl-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  13nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035334((1-Methylsulfanyl-6,7,8,9-tetrahydro-3H-benzo[e]in...)
Affinity DataKi:  13nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035310((1-Methyl-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  14nMAssay Description:Binding affinity against Dopamine receptor D2 expressed in CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035333(1-(8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]i...)
Affinity DataKi:  14nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035317(((R)-4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-...)
Affinity DataKi:  14nMAssay Description:Binding affinity against Dopamine receptor D3 from CHO-K1 cells, using [3H]-spiperone as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035308(8-Dipropylamino-1,3,6,7,8,9-hexahydro-benzo[e]indo...)
Affinity DataKi:  14nMAssay Description:Binding affinity against 5-hydroxytryptamine 1A receptor from CHO-K1 cells, using [3H]-8-OH-DPAT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035317(((R)-4-Fluoro-6,7,8,9-tetrahydro-3H-benzo[e]indol-...)
Affinity DataKi:  14nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035329((+/-)-Dipropyl-(6,7,8,9-tetrahydro-3H-benzo[e]indo...)
Affinity DataKi:  15nMAssay Description:Binding affinity against Dopamine receptor D2 expressed in CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035306((1-Chloro-6,7,8,9-tetrahydro-3H-benzo[e]indol-8-yl...)
Affinity DataKi:  15nMAssay Description:Binding affinity against Dopamine receptor D3 expressed in CHO-K1 cells, using [3H]-spiperone as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1D(Homo sapiens (Human))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035330(CHEMBL302172 | Dipropyl-(R)-6,7,8,9-tetrahydro-3H-...)
Affinity DataKi:  16nMAssay Description:Binding affinity against 5-hydroxytryptamine 1D receptor alpha expressed in CHO-K1 cells, using [3H]-5-HT as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
GöTeborg University

Curated by ChEMBL
LigandPNGBDBM50035303((R)-8-Dipropylamino-6,7,8,9-tetrahydro-3H-benzo[e]...)
Affinity DataKi:  17nMAssay Description:Binding affinity against Dopamine receptor D2 from CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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