TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 0.000320nMAssay Description:Binding affinity kappa opioid receptor in guinea pig brain membranes; using 1 nM [3H]-U69,593 as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataIC50: 2.20nMAssay Description:Binding affinity kappa opioid receptor in guinea pig brain membranes, using 1 nM [3H]-U69,593 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 31nMAssay Description:Binding affinity for mu opioid receptor in guinea pig brain membranes; using 2 nM [3H]-DAMGO as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 89nMAssay Description:Binding affinity for delta opioid receptor in guinea pig brain membranes; using 2 nM [3H]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity for delta opioid receptor in guinea pig brain membranes, using 2 nM [3H]-DPDPE as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.80E+3nMAssay Description:Binding affinity for mu opioid receptor in guinea pig brain membranes, using 2 nM [3H]-DAMGO as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 2.40nMAssay Description:Tested for competitive covalent binding of compound against k opioid receptor in guinea pig brain membrane using [3H]-U-69,593 as radioligandMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota
Curated by ChEMBL
University Of Minnesota
Curated by ChEMBL
Affinity DataKd: 3.40nMAssay Description:Tested for competitive covalent binding of compound against k opioid receptor in guinea pig brain membrane; using [3H]-U-69,593 as radioligandMore data for this Ligand-Target Pair