Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50003379
TargetSubstance-K receptor(Human)
Glaxo Institute For Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50469874(CHEMBL59780)
Affinity DataKi:  0.155nMAssay Description:Binding affinity against human NK2 receptors expressed in CHO cells using [3H]GR-100679 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Glaxo Institute For Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50469872(CHEMBL413650)
Affinity DataKi:  1.30nMAssay Description:Binding affinity against human NK2 receptors expressed in CHO cells using [3H]GR-100679 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Glaxo Institute For Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50469869(CHEMBL217548)
Affinity DataKi:  1.40nMAssay Description:Binding affinity against human NK2 receptors expressed in CHO cells using [3H]GR-100679 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Glaxo Institute For Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50469867(CHEMBL268783)
Affinity DataKi:  1.5nMAssay Description:Binding affinity against human NK2 receptors expressed in CHO cells using [3H]GR-100679 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Glaxo Institute For Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50469870(CHEMBL275499)
Affinity DataKi:  6.60nMAssay Description:Binding affinity against human NK2 receptors expressed in CHO cells using [3H]GR-100679 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Glaxo Institute For Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50469868(CHEMBL413205)
Affinity DataKi:  25nMAssay Description:Binding affinity against human NK2 receptors expressed in CHO cells using [3H]GR-100679 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Glaxo Institute For Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50469871(CHEMBL386783)
Affinity DataKi:  87nMAssay Description:Binding affinity against human NK2 receptors expressed in CHO cells using [3H]GR-100679 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetSubstance-K receptor(Human)
Glaxo Institute For Molecular Biology

Curated by ChEMBL
LigandPNGBDBM50469873(CHEMBL411905)
Affinity DataKi:  1.02E+3nMAssay Description:Binding affinity against human NK2 receptors expressed in CHO cells using [3H]GR-100679 as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed