Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 50005871
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041917BDBM50041917(4-{4-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-phenyl}-2...)
Affinity DataIC50: 10nMAssay Description:In vitro PAF antagonistic activity by determining [3H]PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041919BDBM50041919(6-{4-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-phenyl}-3...)
Affinity DataIC50: 40nMAssay Description:In vitro PAF antagonistic activity by determining [3H]PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041924BDBM50041924(7-Methyl-4-{4-[2-(3,4,5-trimethoxy-phenyl)-ethyl]-...)
Affinity DataIC50: 50nMAssay Description:In vitro PAF antagonistic activity by determining [3H]PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041916BDBM50041916(2,2-Dimethyl-5-{4-[2-(3,4,5-trimethoxy-phenyl)-eth...)
Affinity DataIC50: 60nMAssay Description:In vitro PAF antagonistic activity by determining [3H]PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041921BDBM50041921(SDZ-64-412 | 5-{4-[2-(3,4,5-Trimethoxy-phenyl)-eth...)
Affinity DataIC50: 60nMAssay Description:In vitro PAF antagonistic activity by determining [3H]PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041926BDBM50041926(2-Methyl-5-{4-[2-(3,4,5-trimethoxy-phenyl)-ethyl]-...)
Affinity DataIC50: 220nMAssay Description:In vitro PAF antagonistic activity by determining [3H]PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041923BDBM50041923(3,3-Dimethyl-6-{4-[2-(3,4,5-trimethoxy-phenyl)-eth...)
Affinity DataIC50: 500nMAssay Description:In vitro PAF antagonistic activity by determining [3H]PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041920BDBM50041920(5-{4-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-phenyl}-2...)
Affinity DataIC50: 1.14E+3nMAssay Description:In vitro PAF antagonistic activity by determining [3H]PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041918BDBM50041918(3-Methyl-5-{4-[2-(3,4,5-trimethoxy-phenyl)-ethyl]-...)
Affinity DataIC50: 9.50E+3nMAssay Description:In vitro PAF antagonistic activity by determining [3H]PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041925BDBM50041925(2-Methyl-5-{4-[2-(3,4,5-trimethoxy-phenyl)-ethyl]-...)
Affinity DataIC50: 3.50E+4nMAssay Description:In vitro PAF antagonistic activity by determining [3H]PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPlatelet-activating factor receptor(Human)
Sandoz Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50041922BDBM50041922(5-{4-[2-(3,4,5-Trimethoxy-phenyl)-ethyl]-phenyl}-i...)
Affinity DataIC50: 8.90E+4nMAssay Description:In vitro PAF antagonistic activity by determining [3H]PAF binding to the PAF-receptor of human plateletsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed