Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 50036192
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043326BDBM50043326(c(Cys-Ser-Cys)-Ser-Ser-Leu-Met-Asp-Lys-Gln-c(Cys-V...)
Affinity DataIC50: 0.0930nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000558BDBM50000558(Endothelin-1 | ET-1 | Endothelin -1 | c(Cys-Ser-c(...)
Affinity DataIC50: 0.120nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50000558BDBM50000558(Endothelin-1 | ET-1 | Endothelin -1 | c(Cys-Ser-c(...)
Affinity DataIC50: 0.150nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043322BDBM50043322(c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-V...)
Affinity DataIC50: 0.170nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368776BDBM50368776(CHEMBL1790962)
Affinity DataIC50: 0.170nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368773BDBM50368773(CHEMBL1790959)
Affinity DataIC50: 0.180nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368774BDBM50368774(CHEMBL1790963)
Affinity DataIC50: 0.190nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368775BDBM50368775(CHEMBL1790960)
Affinity DataIC50: 0.200nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368772BDBM50368772(CHEMBL2373291)
Affinity DataIC50: 0.25nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368774BDBM50368774(CHEMBL1790963)
Affinity DataIC50: 0.330nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368777BDBM50368777(CHEMBL2373292)
Affinity DataIC50: 0.420nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368776BDBM50368776(CHEMBL1790962)
Affinity DataIC50: 0.420nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin receptor type B(Bovine)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043324BDBM50043324(c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-V...)
Affinity DataIC50: 0.450nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in bovine cerebrum membrane for Endothelin B receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368772BDBM50368772(CHEMBL2373291)
Affinity DataIC50: 0.700nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50368777BDBM50368777(CHEMBL2373292)
Affinity DataIC50: 0.700nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043322BDBM50043322(c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-V...)
Affinity DataIC50: 0.75nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043326BDBM50043326(c(Cys-Ser-Cys)-Ser-Ser-Leu-Met-Asp-Lys-Gln-c(Cys-V...)
Affinity DataIC50: 5.90nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed
TargetEndothelin-1 receptor(Pig)
Takeda Chemical Industries

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50043324BDBM50043324(c(Cys-Ser-c(Cys-Ser-Ser-Leu-Met-Asp-Lys-Gln-Cys)-V...)
Affinity DataIC50: 8.60nMAssay Description:Tested for the competitive binding versus [125I]- ET-1 determined in porcine cardiac ventricular membrane for Endothelin A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/26/2012
Entry Details Article
PubMed