Compile Data Set for Download or QSAR
maximum 50k data
Found 20 Enz. Inhib. hit(s) with all data for entry = 50006117
TargetMu-type opioid receptor(GUINEA PIG)
University Of California

Curated by ChEMBL
LigandPNGBDBM50140906(1-[2-[1-[2-amino-3-(4-hydroxyphenyl)-(2S)-propanoy...)
Affinity DataIC50:  21nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456337(CHEMBL267708)
Affinity DataIC50:  29nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456336(CHEMBL2371360)
Affinity DataIC50:  31nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456335(CHEMBL2371359)
Affinity DataIC50:  109nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456332(CHEMBL2371339)
Affinity DataIC50:  170nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456336(CHEMBL2371360)
Affinity DataIC50:  202nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of California

Curated by ChEMBL
LigandPNGBDBM50166066(CHEMBL362991 | H-Tyr-Pro-Phe-Pro-NH2 | MORPHICEPTI...)
Affinity DataIC50:  552nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456334(CHEMBL2371340)
Affinity DataIC50:  557nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456335(CHEMBL2371359)
Affinity DataIC50:  594nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of California

Curated by ChEMBL
LigandPNGBDBM50140906(1-[2-[1-[2-amino-3-(4-hydroxyphenyl)-(2S)-propanoy...)
Affinity DataIC50:  1.25E+3nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456337(CHEMBL267708)
Affinity DataIC50:  1.51E+3nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456332(CHEMBL2371339)
Affinity DataIC50:  1.79E+3nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456339(CHEMBL2371336)
Affinity DataIC50:  2.66E+3nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of California

Curated by ChEMBL
LigandPNGBDBM50166066(CHEMBL362991 | H-Tyr-Pro-Phe-Pro-NH2 | MORPHICEPTI...)
Affinity DataIC50:  3.69E+3nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456334(CHEMBL2371340)
Affinity DataIC50:  4.81E+3nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456333(CHEMBL2371361)
Affinity DataIC50:  2.69E+4nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456338(CHEMBL2371337)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory activity against mu opioid receptor using guinea pig ileum (GPI) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456333(CHEMBL2371361)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456339(CHEMBL2371336)
Affinity DataIC50:  5.65E+5nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of California

Curated by ChEMBL
LigandPNGBDBM50456338(CHEMBL2371337)
Affinity DataIC50: >1.00E+6nMAssay Description:In vitro inhibitory activity against delta opioid receptor using mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed