Compile Data Set for Download or QSAR
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Found 7 Enz. Inhib. hit(s) with all data for entry = 50036126
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Monsanto

Curated by ChEMBL
LigandPNGBDBM50046132(2-[propyl-hydroxy-phosphorylamino)-4-methyl-pentan...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of endothelin converting enzyme in an RIA assay using ET-1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Monsanto

Curated by ChEMBL
LigandPNGBDBM50251742((3R,4R,5R,6S)-3,4,5-trihydroxy-6-methyl-tetrahydro...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of endothelin converting enzyme in an RIA assay using ET-1 as substrate (value corresponds to <25% inhibition when assayed at a 100 uM scr...More data for this Ligand-Target Pair
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Monsanto

Curated by ChEMBL
LigandPNGBDBM50046138(2-[2-(Cyclohexylmethyl-hydroxy-phosphorylamino)-4-...)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of endothelin converting enzyme in an RIA assay using ET-1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Monsanto

Curated by ChEMBL
LigandPNGBDBM50046137(2-[2-(Hydroxy-phenoxy-phosphorylamino)-4-methyl-pe...)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of endothelin converting enzyme in an RIA assay using ET-1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Monsanto

Curated by ChEMBL
LigandPNGBDBM50046134(2-[2-(Cyclohexyloxy-hydroxy-phosphorylamino)-4-met...)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibition of endothelin converting enzyme in an RIA assay using ET-1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Monsanto

Curated by ChEMBL
LigandPNGBDBM50046133(2-[2-(Hydroxy-benzyl-phosphorylamino)-4-methyl-pen...)
Affinity DataIC50:  6.10E+4nMAssay Description:Inhibition of endothelin converting enzyme in an RIA assay using ET-1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Monsanto

Curated by ChEMBL
LigandPNGBDBM50046135(2-[2-(Ethoxy-hydroxy-phosphorylamino)-4-methyl-pen...)
Affinity DataIC50:  1.09E+5nMAssay Description:Inhibition of endothelin converting enzyme in an RIA assay using ET-1 as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed