Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with all data for entry = 50006352
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50005576((3S,8R)-3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3...)
Affinity DataIC50:  1.60nMAssay Description:Compounds binding ability to dopamine transporter was evaluated by displacing [3H]-beta-CFT in baboon brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Northeastern University

Curated by ChEMBL
LigandPNGBDBM50005576((3S,8R)-3-(4-Iodo-phenyl)-8-methyl-8-aza-bicyclo[3...)
Affinity DataIC50:  3.80nMAssay Description:Compounds binding ability to serotonin transporter was evaluated by displacing [3H]-paroxetine in baboon brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed