Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50038916
TargetcAMP-dependent protein kinase(Rabbit)
Institute For Biochemistry

Curated by ChEMBL
LigandPNGBDBM15210(N-[2-(methylamino)ethyl]isoquinoline-5-sulfonamide...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibitory constant against cAPK (PKA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetcAMP-dependent protein kinase(Rabbit)
Institute For Biochemistry

Curated by ChEMBL
LigandPNGBDBM50366348(CHEMBL1233654)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibitory constant against cAPK (PKA)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetMyosin light chain kinase, smooth muscle(Chicken)
Institute For Biochemistry

Curated by ChEMBL
LigandPNGBDBM15211(CHEMBL104264 | H89 | N-(2-{[(2E)-3-(4-bromophenyl)...)
Affinity DataKi:  2.83E+4nMAssay Description:Inhibitory constant against MLCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetMyosin light chain kinase, smooth muscle(Chicken)
Institute For Biochemistry

Curated by ChEMBL
LigandPNGBDBM15210(N-[2-(methylamino)ethyl]isoquinoline-5-sulfonamide...)
Affinity DataKi:  6.80E+4nMAssay Description:Inhibitory constant against MLCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetMyosin light chain kinase, smooth muscle(Chicken)
Institute For Biochemistry

Curated by ChEMBL
LigandPNGBDBM50366348(CHEMBL1233654)
Affinity DataKi:  9.70E+4nMAssay Description:Inhibitory constant against MLCKMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha (Human)
Institute For Biochemistry

Curated by ChEMBL
LigandPNGBDBM15211(CHEMBL104264 | H89 | N-(2-{[(2E)-3-(4-bromophenyl)...)
Affinity DataKi:  1.37E+5nMAssay Description:Inhibitory constant against bovine CK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha (Human)
Institute For Biochemistry

Curated by ChEMBL
LigandPNGBDBM50366348(CHEMBL1233654)
Affinity DataKi:  7.80E+5nMAssay Description:Inhibitory constant against CK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed
TargetCasein kinase II subunit alpha (Human)
Institute For Biochemistry

Curated by ChEMBL
LigandPNGBDBM15210(N-[2-(methylamino)ethyl]isoquinoline-5-sulfonamide...)
Affinity DataKi:  9.50E+5nMAssay Description:Inhibitory constant against CK2More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/24/2012
Entry Details Article
PubMed