Compile Data Set for Download or QSAR
Report error Found 207 Enz. Inhib. hit(s) with all data for entry = 8907
TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427431BDBM427431(US10544136, Compound 215 | US10544136, Compound 21...)
Affinity DataEC50:  0.100nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427424BDBM427424(US10544136, Compound 209)
Affinity DataEC50:  0.140nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427221BDBM427221(US10544136, Compound 32)
Affinity DataEC50:  0.150nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427392BDBM427392(US10544136, Compound 123)
Affinity DataEC50:  0.200nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427476BDBM427476(US10544136, Compound 262)
Affinity DataEC50: <0.5nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427474BDBM427474(US10544136, Compound 261)
Affinity DataEC50: <0.5nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427473BDBM427473(US10544136, Compound 260)
Affinity DataEC50: <0.5nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427472BDBM427472(US10544136, Compound 259)
Affinity DataEC50: <0.5nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 429762BDBM429762(US10544136, Compound 271)
Affinity DataEC50: <0.5nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427450BDBM427450(US10544136, Compound 234)
Affinity DataEC50: <0.5nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427481BDBM427481(US10544136, Compound 265)
Affinity DataEC50: <0.5nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427417BDBM427417(US10544136, Compound 201)
Affinity DataEC50:  0.5nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427389BDBM427389(US10544136, Compound 110)
Affinity DataEC50:  0.520nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427461BDBM427461(US10544136, Compound 243)
Affinity DataEC50:  0.700nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427252BDBM427252(US10544136, Compound 61)
Affinity DataEC50:  0.780nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427406BDBM427406(US10544136, Compound 177)
Affinity DataEC50:  0.800nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427471BDBM427471(US10544136, Compound 258)
Affinity DataEC50:  1nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427251BDBM427251(US10544136, Compound 60)
Affinity DataEC50:  1nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427415BDBM427415(US10544136, Compound 192)
Affinity DataEC50:  1.10nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427452BDBM427452(US10544136, Compound 236)
Affinity DataEC50:  1.10nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427462BDBM427462(US10544136, Compound 248 | US10544136, Compound 25...)
Affinity DataEC50:  1.5nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427402BDBM427402(US10544136, Compound 155)
Affinity DataEC50:  1.70nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427226BDBM427226(US10544136, Compound 36)
Affinity DataEC50:  1.70nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427405BDBM427405(US10544136, Compound 167)
Affinity DataEC50:  2.20nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 429732BDBM429732(US10544136, Compound 270)
Affinity DataEC50:  2.5nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427442BDBM427442(US10544136, Compound 226)
Affinity DataEC50:  2.70nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427393BDBM427393(US10544136, Compound 124)
Affinity DataEC50:  3nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427401BDBM427401(US10544136, Compound 154)
Affinity DataEC50:  3.10nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427212BDBM427212(US10544136, Compound 16)
Affinity DataEC50:  3.30nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427465BDBM427465(US10544136, Compound 251)
Affinity DataEC50:  3.40nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 37115BDBM37115(5-(3,4-diethoxyphenyl)-3-pyridin-4-yl-1,2,4-oxadia...)
Affinity DataEC50:  3.70nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427396BDBM427396(US10544136, Compound 129)
Affinity DataEC50:  4.10nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427411BDBM427411(US10544136, Compound 186)
Affinity DataEC50:  4.20nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427397BDBM427397(US10544136, Compound 150)
Affinity DataEC50:  4.20nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427391BDBM427391(US10544136, Compound 122)
Affinity DataEC50:  5nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427253BDBM427253(US10544136, Compound 62)
Affinity DataEC50:  5nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427398BDBM427398(US10544136, Compound 151)
Affinity DataEC50:  5.90nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427399BDBM427399(US10544136, Compound 152)
Affinity DataEC50:  6nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427462BDBM427462(US10544136, Compound 248 | US10544136, Compound 25...)
Affinity DataEC50:  6.10nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427400BDBM427400(US10544136, Compound 153)
Affinity DataEC50:  6.90nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427413BDBM427413(US10544136, Compound 187)
Affinity DataEC50:  7nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 36953BDBM36953(MLS000042464 | cid_666359 | 3-(3,4-diethoxyphenyl)...)
Affinity DataEC50:  7.30nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427480BDBM427480(US10544136, Compound 264)
Affinity DataEC50:  8nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427224BDBM427224(US10544136, Compound 34)
Affinity DataEC50:  8.80nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427479BDBM427479(US10544136, Compound 263)
Affinity DataEC50:  10nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427467BDBM427467(US10544136, Compound 252)
Affinity DataEC50:  10.1nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 429591BDBM429591(US10544136, Compound 268)
Affinity DataEC50:  10.7nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427250BDBM427250(US10544136, Compound 59)
Affinity DataEC50:  10.8nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427408BDBM427408(US10544136, Compound 184)
Affinity DataEC50:  11.7nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
The Scripps Research Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 427249BDBM427249(US10544136, Compound 58)
Affinity DataEC50:  11.7nMAssay Description:The method involves contacting the receptor with a suitable concentration of an inventive compound to bring about activation of the receptor. The con...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2020
Entry Details
US Patent

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