Compile Data Set for Download or QSAR
maximum 50k data
Found 33 Enz. Inhib. hit(s) with all data for entry = 50036591
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454823(CHEMBL3084910)
Affinity DataKi:  0.410nMAssay Description:Displacement of [3H]pirenzepine binding at muscarinic Muscarinic acetylcholine receptor M1 in rat brain P2 membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454830(CHEMBL3084869)
Affinity DataKi:  0.430nMAssay Description:Displacement of [3H]pirenzepine binding at muscarinic Muscarinic acetylcholine receptor M1 in rat brain P2 membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454825(CHEMBL3084878)
Affinity DataKi:  0.5nMAssay Description:Displacement of [3H]pirenzepine binding at muscarinic Muscarinic acetylcholine receptor M1 in rat brain P2 membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50366775(BENZTROPINE | Benzatropine)
Affinity DataKi:  0.590nMAssay Description:Displacement of [3H]pirenzepine binding at muscarinic Muscarinic acetylcholine receptor M1 in rat brain P2 membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454828(CHEMBL3084907)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]pirenzepine binding at muscarinic Muscarinic acetylcholine receptor M1 in rat brain P2 membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454824(CHEMBL3084909)
Affinity DataKi:  0.850nMAssay Description:Displacement of [3H]pirenzepine binding at muscarinic Muscarinic acetylcholine receptor M1 in rat brain P2 membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454829(CHEMBL3084870)
Affinity DataKi:  0.980nMAssay Description:Displacement of [3H]pirenzepine binding at muscarinic Muscarinic acetylcholine receptor M1 in rat brain P2 membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454827(AMINOBENZTROPINE)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]pirenzepine binding at muscarinic Muscarinic acetylcholine receptor M1 in rat brain P2 membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM86702(3-[(4-Chloro-phenyl)-phenyl-methoxy]-8-methyl-8-az...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]pirenzepine binding at muscarinic Muscarinic acetylcholine receptor M1 in rat brain P2 membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(RAT)
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454826(CHEMBL3084901)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]pirenzepine binding at muscarinic Muscarinic acetylcholine receptor M1 in rat brain P2 membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454829(CHEMBL3084870)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]WIN-35428 binding to the dopamine transporter (DAT) in Rat Caudate PutamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM86702(3-[(4-Chloro-phenyl)-phenyl-methoxy]-8-methyl-8-az...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]WIN-35428 binding to the dopamine transporter (DAT) in Rat Caudate PutamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]WIN-35428 binding to the dopamine transporter (DAT) in Rat Caudate PutamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataKi:  32nMAssay Description:Displacement of [3H]WIN-35428 binding to the dopamine transporter (DAT) in Rat Caudate PutamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454824(CHEMBL3084909)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]WIN-35428 binding to the dopamine transporter (DAT) in Rat Caudate PutamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454830(CHEMBL3084869)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]WIN-35428 binding to the dopamine transporter (DAT) in Rat Caudate PutamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454828(CHEMBL3084907)
Affinity DataKi:  69nMAssay Description:Displacement of [3H]WIN-35428 binding to the dopamine transporter (DAT) in Rat Caudate PutamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50366775(BENZTROPINE | Benzatropine)
Affinity DataKi:  118nMAssay Description:Displacement of [3H]WIN-35428 binding to the dopamine transporter (DAT) in Rat Caudate PutamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454826(CHEMBL3084901)
Affinity DataKi:  187nMAssay Description:Displacement of [3H]WIN-35428 binding to the dopamine transporter (DAT) in Rat Caudate PutamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454823(CHEMBL3084910)
Affinity DataKi:  228nMAssay Description:Displacement of [3H]WIN-35428 binding to the dopamine transporter (DAT) in Rat Caudate PutamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454825(CHEMBL3084878)
Affinity DataKi:  309nMAssay Description:Displacement of [3H]WIN-35428 binding to the dopamine transporter (DAT) in Rat Caudate PutamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454827(AMINOBENZTROPINE)
Affinity DataKi:  1.84E+3nMAssay Description:Displacement of [3H]WIN-35428 binding to the dopamine transporter (DAT) in Rat Caudate PutamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50084717((+)-(1R,2R,3S,5S)-methyl 3-(benzoyloxy)-8-methyl-8...)
Affinity DataIC50:  12nMAssay Description:[3H]-Dopamine uptake inhibition in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM86702(3-[(4-Chloro-phenyl)-phenyl-methoxy]-8-methyl-8-az...)
Affinity DataIC50:  115nMAssay Description:[3H]-Dopamine uptake inhibition in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454830(CHEMBL3084869)
Affinity DataIC50:  140nMAssay Description:[3H]-Dopamine uptake inhibition in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454829(CHEMBL3084870)
Affinity DataIC50:  228nMAssay Description:[3H]-Dopamine uptake inhibition in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454828(CHEMBL3084907)
Affinity DataIC50:  250nMAssay Description:[3H]-Dopamine uptake inhibition in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454827(AMINOBENZTROPINE)
Affinity DataIC50:  373nMAssay Description:[3H]-Dopamine uptake inhibition in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50366775(BENZTROPINE | Benzatropine)
Affinity DataIC50:  403nMAssay Description:[3H]-Dopamine uptake inhibition in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454824(CHEMBL3084909)
Affinity DataIC50:  407nMAssay Description:[3H]-Dopamine uptake inhibition in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454826(CHEMBL3084901)
Affinity DataIC50:  457nMAssay Description:[3H]-Dopamine uptake inhibition in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454823(CHEMBL3084910)
Affinity DataIC50:  997nMAssay Description:[3H]-Dopamine uptake inhibition in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
National Institutes Of Health

Curated by ChEMBL
LigandPNGBDBM50454825(CHEMBL3084878)
Affinity DataIC50:  1.20E+3nMAssay Description:[3H]-Dopamine uptake inhibition in rat caudate putamenMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed