Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with all data for entry = 50007565
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064703((R)-2-(8-Bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-...)
Affinity DataKi:  0.300nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2C receptor using [125 I]DOI as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064703((R)-2-(8-Bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-...)
Affinity DataKi:  0.480nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2A receptor using [125 I]DOI as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064703((R)-2-(8-Bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-...)
Affinity DataKi:  1.15nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2B receptor using [3H]-rauwolscine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064703((R)-2-(8-Bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-...)
Affinity DataKi:  1.60nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT 2B as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064703((R)-2-(8-Bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-...)
Affinity DataKi:  2.28nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2C receptor using [3H]- mesulergine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064706((2aS,4R)-8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-...)
Affinity DataKi:  5.96nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2C receptor using [125 I]DOI as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064703((R)-2-(8-Bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-...)
Affinity DataKi:  11nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2A receptor using [3H]-ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064706((2aS,4R)-8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-...)
Affinity DataKi:  13nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2A receptor using [125 I]DOI as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064703((R)-2-(8-Bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-...)
Affinity DataKi:  18nMAssay Description:Affinity at [3H]-ketanserin-labeled 5-hydroxytryptamine 2A receptor in rat brain homogenate was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064708((R)-1-(4-bromo-2,5-dimethoxyphenyl)propan-2-amine ...)
Affinity DataKi:  22nMAssay Description:Affinity at [3H]-ketanserin-labeled 5-hydroxytryptamine 2A receptor in rat brain homogenate was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064706((2aS,4R)-8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-...)
Affinity DataKi:  90nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2C receptor using [3H]- mesulergine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064706((2aS,4R)-8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-...)
Affinity DataKi:  240nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2A receptor using [3H]-ketanserin as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064706((2aS,4R)-8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-...)
Affinity DataKi:  255nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2B receptor using [3H]- rauwolscine as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064706((2aS,4R)-8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-...)
Affinity DataKi:  263nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT 2B as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064704(((2aS,4R)-6-Methoxy-2a,3,4,5-tetrahydro-2H-naphtho...)
Affinity DataKi:  644nMAssay Description:Affinity at [3H]-ketanserin-labeled 5-hydroxytryptamine 2A receptor in rat brain homogenate was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064707(((2aS,4R)-6-Methoxy-2a,3,4,5-tetrahydro-2H-naphtho...)
Affinity DataKi:  967nMAssay Description:Affinity at [3H]-ketanserin-labeled 5-hydroxytryptamine 2A receptor in rat brain homogenate was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064706((2aS,4R)-8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-...)
Affinity DataKi:  1.05E+3nMAssay Description:Affinity at [3H]-ketanserin-labeled 5-hydroxytryptamine 2A receptor in rat brain homogenate was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064705((2aR,4R)-8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-...)
Affinity DataKi:  3.88E+3nMAssay Description:Affinity at [3H]-ketanserin-labeled 5-hydroxytryptamine 2A receptor in rat brain homogenate was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064705((2aR,4R)-8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-...)
Affinity DataKi:  4.19E+3nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2C receptor using [125 I]DOI as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064703((R)-2-(8-Bromo-2,3,6,7-tetrahydro-benzo[1,2-b;4,5-...)
Affinity DataKi:  4.30E+3nMAssay Description:Affinity at [3H]-8-OH-DPAT-labeled 5-hydroxytryptamine 1A receptor in rat brain homogenate was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064708((R)-1-(4-bromo-2,5-dimethoxyphenyl)propan-2-amine ...)
Affinity DataKi:  6.10E+3nMAssay Description:Affinity at [3H]-8-OH-DPAT-labeled 5-hydroxytryptamine 1A receptor in rat brain homogenate was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064705((2aR,4R)-8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-...)
Affinity DataKi:  8.50E+3nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2A receptor using [125 I]DOI as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064705((2aR,4R)-8-Bromo-6-methoxy-2a,3,4,5-tetrahydro-2H-...)
Affinity DataKi:  1.12E+4nMAssay Description:Binding ability of compound at cloned human 5-hydroxytryptamine 2B receptor using [3H]-5-HT 2B as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064707(((2aS,4R)-6-Methoxy-2a,3,4,5-tetrahydro-2H-naphtho...)
Affinity DataKi:  3.80E+4nMAssay Description:Affinity at [3H]-8-OH-DPAT-labeled 5-hydroxytryptamine 1A receptor in rat brain homogenate was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Purdue University

Curated by ChEMBL
LigandPNGBDBM50064704(((2aS,4R)-6-Methoxy-2a,3,4,5-tetrahydro-2H-naphtho...)
Affinity DataKi:  1.44E+5nMAssay Description:Affinity at [3H]-8-OH-DPAT-labeled 5-hydroxytryptamine 1A receptor in rat brain homogenate was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed