Compile Data Set for Download or QSAR
Report error Found 14 Enz. Inhib. hit(s) with all data for entry = 50041022
Target5-hydroxytryptamine receptor 1A(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50026917(CHEMBL13647 | BMY 7378 | 8-{2-[4-(2-Methoxy-phenyl...)
Affinity DataKi:  1.70nMAssay Description:Antagonistic affinity against cloned human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50026917(CHEMBL13647 | BMY 7378 | 8-{2-[4-(2-Methoxy-phenyl...)
Affinity DataKi:  48nMAssay Description:Antagonistic affinity against rat striatum Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
LigandPNGBDBM50403647(CHEMBL27013)
Affinity DataKi:  100nMAssay Description:Antagonistic affinity against native rat cortex Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi:  158nMAssay Description:Antagonistic affinity against native rat cortex Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
LigandPNGBDBM50403651(CHEMBL29591)
Affinity DataKi:  589nMAssay Description:Antagonistic affinity against native rat cortex Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
LigandPNGBDBM50403649(CYCLAZOSIN)
Affinity DataKi:  741nMAssay Description:Antagonistic affinity against native rat cortex Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50403647(CHEMBL27013)
Affinity DataKi: <1.00E+3nMAssay Description:Antagonistic affinity against cloned human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50403651(CHEMBL29591)
Affinity DataKi: <1.00E+3nMAssay Description:Antagonistic affinity against cloned human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi: <1.00E+3nMAssay Description:Antagonistic affinity against cloned human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
Target5-hydroxytryptamine receptor 1A(Human)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50403649(CYCLAZOSIN)
Affinity DataKi: <1.00E+3nMAssay Description:Antagonistic affinity against cloned human 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
LigandPNGBDBM50026917(CHEMBL13647 | BMY 7378 | 8-{2-[4-(2-Methoxy-phenyl...)
Affinity DataKi:  1.05E+3nMAssay Description:Antagonistic affinity against native rat cortex Alpha-2 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50403647(CHEMBL27013)
Affinity DataKi:  2.34E+3nMAssay Description:Antagonistic affinity against rat striatum Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM50403649(CYCLAZOSIN)
Affinity DataKi:  8.32E+3nMAssay Description:Antagonistic affinity against rat striatum Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed
TargetD(2) dopamine receptor(Rat)
University of Bologna

Curated by ChEMBL
LigandPNGBDBM29568([3H]-Minipress | [3H]-Furazosin | PRAZOSIN HYDROCH...)
Affinity DataKi: <1.00E+4nMAssay Description:Antagonistic affinity against rat striatum Dopamine receptor D2More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article
PubMed