Compile Data Set for Download or QSAR
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Found 28 Enz. Inhib. hit(s) with all data for entry = 50008066
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070420((2S,4S)-1-[(S)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  14nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070414(CHEMBL286247 | {[(R)-2-(Adamantan-2-yloxycarbonyla...)
Affinity DataKi:  14nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070412((2R,4R)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  15nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataKi:  15nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070415((2R,4R)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  19nMAssay Description:Inhibitory activity against CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070413((2R,4R)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  24nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070419((2R,4R)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  28nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070416((2R,4R)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  33nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070411((2R,4S)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  175nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070424((2S,4R)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  543nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070412((2R,4R)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  751nMAssay Description:Binding affinity against CCK-A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070417((2R,4R)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  789nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070423((2S,4S)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  791nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070418((2R,4S)-1-[(S)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  812nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070421((2S,4R)-1-[(S)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  896nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50450641(CHEMBL2114379)
Affinity DataKi:  1.04E+3nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070420((2S,4S)-1-[(S)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  1.06E+3nMAssay Description:Binding affinity against CCK-A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070414(CHEMBL286247 | {[(R)-2-(Adamantan-2-yloxycarbonyla...)
Affinity DataKi:  1.06E+3nMAssay Description:Binding affinity against CCK-A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070422((2R,4S)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  1.54E+3nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070410(CHEMBL105618 | [2-(4-Benzoyl-piperidin-1-yl)-1-(1H...)
Affinity DataKi:  1.70E+3nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070410(CHEMBL105618 | [2-(4-Benzoyl-piperidin-1-yl)-1-(1H...)
Affinity DataKi:  1.70E+3nMAssay Description:Binding affinity against CCK-A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCholecystokinin receptor type A(Cavia porcellus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070411((2R,4S)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataKi:  3.72E+3nMAssay Description:Binding affinity against CCK-A receptor in guinea pig pancreatic membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070412((2R,4R)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataIC50:  37nMAssay Description:Inhibitory activity against CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50006878((R)-1-(1-Methyl-2-oxo-5-phenyl-2,3-dihydro-1H-benz...)
Affinity DataIC50:  39nMAssay Description:Inhibitory activity against CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070420((2S,4S)-1-[(S)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataIC50:  217nMAssay Description:Inhibitory activity against CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070414(CHEMBL286247 | {[(R)-2-(Adamantan-2-yloxycarbonyla...)
Affinity DataIC50:  217nMAssay Description:Capacity to inhibit [3H]-p CCK 8 binding to membrane preparations of CHO cells transfected with the rat CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070415((2R,4R)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataIC50:  389nMAssay Description:Inhibitory activity against CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50070416((2R,4R)-1-[(R)-2-(Adamantan-2-yloxycarbonylamino)-...)
Affinity DataIC50:  507nMAssay Description:Inhibitory activity against CCK-B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed