Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 50034937
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070679BDBM50070679((S)-2-[(S)-2-{(S)-3-(4-Fluoro-phenyl)-2-[(E)-(3-ph...)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070674BDBM50070674(2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-acetyl...)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070676BDBM50070676(2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-acetyl...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070677BDBM50070677(2-[(S)-1-(2-Amino-3-methyl-butyrylamino)-2-(4-fluo...)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50366502BDBM50366502(CHEMBL1790240)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070673BDBM50070673(2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-acetyl...)
Affinity DataIC50: 4.10E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070656BDBM50070656(2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-acetyl...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070670BDBM50070670(2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-acetyl...)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070669BDBM50070669(2-[(S)-1-(2-Amino-acetylamino)-2-(4-fluoro-phenyl)...)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070672BDBM50070672(2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-acetyl...)
Affinity DataIC50: 5.60E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070657BDBM50070657(2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-acetyl...)
Affinity DataIC50: 5.70E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070654BDBM50070654(2-[(S)-1-(2-Amino-acetylamino)-2-(4-fluoro-phenyl)...)
Affinity DataIC50: 6.20E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070675BDBM50070675(2-[(S)-1-(3-Amino-propionylamino)-2-(4-fluoro-phen...)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070663BDBM50070663(2-[(S)-1-Amino-2-(4-fluoro-phenyl)-ethyl]-thiazole...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070667BDBM50070667(2-[(S)-1-(2-Amino-3-methyl-butyrylamino)-2-(4-meth...)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070658BDBM50070658(2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-acetyl...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070661BDBM50070661(2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-acetyl...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070666BDBM50070666(2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-acetyl...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070665BDBM50070665(2-[(S)-1-Acetylamino-2-(4-fluoro-phenyl)-ethyl]-5-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070671BDBM50070671(2-[(S)-1-(2,3-Diamino-propionylamino)-2-(4-fluoro-...)
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070678BDBM50070678(5-Methyl-2-[(S)-1-(2-methylamino-acetylamino)-2-ph...)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50031392BDBM50031392((S)-2-[(S)-2-((S)-2-{(S)-2-[(S)-2-((S)-2-Amino-3-h...)
Affinity DataIC50: 7.30E+4nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070664BDBM50070664(2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-acetyl...)
Affinity DataIC50: 9.40E+4nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070655BDBM50070655(1-{2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-ace...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070660BDBM50070660(2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-acetyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50070659BDBM50070659(2-[(S)-2-(4-Fluoro-phenyl)-1-(2-methylamino-acetyl...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed
TargetProteinase-activated receptor 1(Human)
R. W. Johnson Pharmaceutical Research Institute

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50366501BDBM50366501(CHEMBL1790239)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of [3H]S-(p-F-Phe)-Har-L-Har-KY-NH2 binding to a thrombin receptor (PAR-1) membrane preparation.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2012
Entry Details Article
PubMed