Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50008145
TargetIntegrase(Human immunodeficiency virus type 1)
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50071060(Disodium; [4-(6-amino-imidazo[4,5-h]quinazolin-1-y...)
Affinity DataIC50: 5.30E+4nMAssay Description:Inhibitory activity against HIV integrase in the strand transfer stepMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50071062(Disodium; [4-(8-amino-imidazo[4,5-g]quinazolin-3-y...)
Affinity DataIC50: 6.80E+4nMAssay Description:Inhibitory activity against HIV integrase in the strand transfer stepMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50071060(Disodium; [4-(6-amino-imidazo[4,5-h]quinazolin-1-y...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against HIV integrase in the 3' processing stepMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50071061(Disodium; [5-(8-amino-3H-imidazo[4,5-g]quinazolin-...)
Affinity DataIC50: 5.50E+5nMAssay Description:Inhibitory activity against HIV integrase in the strand transfer stepMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetIntegrase(Human immunodeficiency virus type 1)
University of Iowa

Curated by ChEMBL
LigandPNGBDBM50071061(Disodium; [5-(8-amino-3H-imidazo[4,5-g]quinazolin-...)
Affinity DataIC50: 7.50E+5nMAssay Description:Inhibitory activity against HIV integrase in the 3' processing stepMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed