Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with all data for entry = 50008174
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50071242(Acetic acid (6aR,6bS,9S,10aR,12aS)-5-hydroxy-1,3-d...)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of human recombinant farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50071241(Acetic acid (6aR,6bS,9S,10aR,12aS)-5-hydroxy-6b,10...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human recombinant farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50071240(Acetic acid (3S,4aR,6aS,12aR,12bS)-11-hydroxy-8,9-...)
Affinity DataIC50:  4.60E+5nMAssay Description:Inhibition of human recombinant farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50071239(Acetic acid (3S,4aR,6aS,12aR,12bS)-8,9-diformyl-11...)
Affinity DataIC50:  5.60E+5nMAssay Description:Inhibition of human recombinant farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed