Compile Data Set for Download or QSAR
Report error Found 136 Enz. Inhib. hit(s) with all data for entry = 3469
TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401411BDBM401411(US10005768, Compound 25 | 6-(4-(4-cyano-2-(2-metho...)
Affinity DataIC50: 39nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401416BDBM401416(US10005768, Compound 30 | 6-(4-(2-(pyrrolidin-1-yl...)
Affinity DataIC50: 49nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401412BDBM401412(US10005768, Compound 26 | 6-(4-(4-cyano-3-(pyridin...)
Affinity DataIC50: 54nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401489BDBM401489(US10005768, Compound 117 | 6-(4-(2- ((ethyl(methyl...)
Affinity DataIC50: 66nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401403BDBM401403(US10005768, Compound 17 | 6-(4-(4-cyano-2-(1-methy...)
Affinity DataIC50: 67nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401507BDBM401507(US10005768, Compound 122 | (S)-6-(1,2-dihydroxyeth...)
Affinity DataIC50: 79nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401435BDBM401435(US10005768, Compound 49 | 6-(4-(2-(piperidin-1-ylm...)
Affinity DataIC50: 96nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401414BDBM401414(US10005768, Compound 28 | 6-(4-(2-(pyridin-4-yl)-4...)
Affinity DataIC50: 101nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401402BDBM401402(US10005768, Compound 16 | 6-(4-(4-cyano-2-(pyridin...)
Affinity DataIC50: 104nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401431BDBM401431(US10005768, Compound 45 | 6-(4-(2-((3,3-difluoropy...)
Affinity DataIC50: 113nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401415BDBM401415(US10005768, Compound 29 | 6-(4-(2-(pyridin-3-yl)-4...)
Affinity DataIC50: 117nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401490BDBM401490(US10005768, Compound 118 | 6-(4-(2-((diethylamino)...)
Affinity DataIC50: 118nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401406BDBM401406(US10005768, Compound 20 | 6-(4-(4-cyano-2-(6- meth...)
Affinity DataIC50: 124nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401461BDBM401461(US10005768, Compound 87 | 6-(3-chloro-4-(4-fluorop...)
Affinity DataIC50: 128nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401421BDBM401421(US10005768, Compound 35 | 6-(4-(2-((3-oxopiperazin...)
Affinity DataIC50: 141nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401505BDBM401505(US10005768, Compound 164 | 6-(4-(2-(diethylcarbamo...)
Affinity DataIC50: 143nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401401BDBM401401(US10005768, Compound 15 | 6-(4-(4-cyano-2-(pyridin...)
Affinity DataIC50: 147nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401508BDBM401508(US10005768, Compound 123 | 6-(4-(2-(1-methyl-1H-py...)
Affinity DataIC50: 149nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401410BDBM401410(US10005768, Compound 24 | 6-(4-(4-cyano-2-(2- meth...)
Affinity DataIC50: 152nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401442BDBM401442(US10005768, Compound 56 | 6-(4-(3-(pyrrolidin-1-yl...)
Affinity DataIC50: 173nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401480BDBM401480(US10005768, Compound 107 | (S)-1-(6-(4-(2-(piperid...)
Affinity DataIC50: 174nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401441BDBM401441(US10005768, Compound 55 | 6-(4-(4-(trifluoromethyl...)
Affinity DataIC50: 174nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401425BDBM401425(US10005768, Compound 39 | 6-(4-(2-((dimethylamino)...)
Affinity DataIC50: 179nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401499BDBM401499(US10005768, Compound 158 | 6-(4-(2-(1-hydroxy-2-ox...)
Affinity DataIC50: 214nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401419BDBM401419(US10005768, Compound 33 | 6-(4-(2-((4-methylpipera...)
Affinity DataIC50: 221nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401429BDBM401429(US10005768, Compound 43 | 6-(4-(2-(morpholinomethy...)
Affinity DataIC50: 223nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401443BDBM401443(US10005768, Compound 58 | 6-(4-(2-(1-(pyrrolidin-1...)
Affinity DataIC50: 231nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401485BDBM401485(US10005768, Compound 113 | (S)-2-(4-(6-(1,2- dihyd...)
Affinity DataIC50: 249nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401473BDBM401473(US10005768, Compound 100 | 6-(4'-chloro-6-(4-fluor...)
Affinity DataIC50: 276nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401481BDBM401481(US10005768, Compound 108 | 6-(4-(2-((cyclopentylam...)
Affinity DataIC50: 280nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401408BDBM401408(US10005768, Compound 22 | 6-(4-(4-cyano-2-(1-methy...)
Affinity DataIC50: 285nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401511BDBM401511(US10005768, Compound 126 | (S)-2-(4-(2-(1-methyl-1...)
Affinity DataIC50: 288nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401520BDBM401520(US10005768, Compound 135 | (S)-4-(1,2-dihydroxythy...)
Affinity DataIC50: 294nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401447BDBM401447(US10005768, Compound 62 | 6-(4-(3-((3-aminoazetidi...)
Affinity DataIC50: 310nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401510BDBM401510(US10005768, Compound 125 | 2-(4-(2-(1-methyl-1H-py...)
Affinity DataIC50: 311nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401476BDBM401476(US10005768, Compound 103 | 6-(4-(4-fluorophenoxy)-...)
Affinity DataIC50: 312nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401405BDBM401405(US10005768, Compound 19 | 6-(4-(4-cyano-2-(thiophe...)
Affinity DataIC50: 337nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401448BDBM401448(US10005768, Compound 63 | 6-(4-(2-(1-hydroxy-2-nit...)
Affinity DataIC50: 337nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401478BDBM401478(US10005768, Compound 105 | 6-(3-((4-cyanophenoxy)m...)
Affinity DataIC50: 362nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401440BDBM401440(US10005768, Compound 54 | (S)-6-(4-(3-((3-hydroxy-...)
Affinity DataIC50: 366nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401509BDBM401509(US10005768, Compound 124 | 2-(6-carbmoyl-2-(4-(2- ...)
Affinity DataIC50: 367nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401439BDBM401439(US10005768, Compound 53 | 6-(4-(3-(azetidin-1-ylme...)
Affinity DataIC50: 384nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401519BDBM401519(US10005768, Compound 134 | (S)-6-((1-amino-1-oxopr...)
Affinity DataIC50: 393nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401404BDBM401404(US10005768, Compound 18 | 6-(4-((4'-amino-5-cyano-...)
Affinity DataIC50: 426nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401422BDBM401422(US10005768, Compound 36 | (S)-6-(4-(2-((3- hydroxy...)
Affinity DataIC50: 432nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401526BDBM401526(US10005768, Compound 141 | (S)-2-(4-(4-chloro-2-(1...)
Affinity DataIC50: 450nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401487BDBM401487(US10005768, Compound 115 | (R)-1-(2-(4-(2-(pyrroli...)
Affinity DataIC50: 455nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401479BDBM401479(US10005768, Compound 106 | 6-(4-(3-((3-oxopiperazi...)
Affinity DataIC50: 455nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401512BDBM401512(US10005768, Compound 127 | 6-(2-(1H-imidazol-1-yl)...)
Affinity DataIC50: 486nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandChemical structure of BindingDB Monomer ID 401460BDBM401460(US10005768, Compound 86 | 6-(2-chloro-4-(4-fluorop...)
Affinity DataIC50: 490nMAssay Description:The assay buffer was formulated by removing 120 mL from a 1 L bottle of fresh, sterile dH2O (Mediatech, Herndon, Va.) and adding 100 mL of 10×HBSS th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/18/2020
Entry Details
US Patent

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