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Report error Found 105 Enz. Inhib. hit(s) with all data for entry = 538
TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277250(US10072005, Example 43)
Affinity DataEC50:  10nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277290(US10072005, Example 83)
Affinity DataEC50:  10nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277276(US10072005, Example 69)
Affinity DataEC50:  10nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277220(US10072005, Example 13)
Affinity DataEC50:  12.6nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277273(US10072005, Example 66)
Affinity DataEC50:  12.6nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277291(US10072005, Example 84)
Affinity DataEC50:  12.6nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277278(US10072005, Example 71)
Affinity DataEC50:  12.6nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277294(US10072005, Example 87)
Affinity DataEC50:  12.6nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277280(US10072005, Example 73)
Affinity DataEC50:  12.6nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277267(US10072005, Example 60)
Affinity DataEC50:  15.8nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277285(US10072005, Example 78)
Affinity DataEC50:  15.8nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277289(US10072005, Example 82)
Affinity DataEC50:  15.8nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277279(US10072005, Example 72)
Affinity DataEC50:  15.8nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277217(US10072005, Example 10)
Affinity DataEC50:  20nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277265(US10072005, Example 58)
Affinity DataEC50:  20nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277219(US10072005, Example 12)
Affinity DataEC50:  20nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277272(US10072005, Example 65)
Affinity DataEC50:  20nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277275(US10072005, Example 68)
Affinity DataEC50:  20nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277254(US10072005, Example 47 | US10072005, Example 48)
Affinity DataEC50:  25.1nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277270(US10072005, Example 63)
Affinity DataEC50:  25.1nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277293(US10072005, Example 86)
Affinity DataEC50:  25.1nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277264(US10072005, Example 57)
Affinity DataEC50:  25.1nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277252(US10072005, Example 45)
Affinity DataEC50:  31.6nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277274(US10072005, Example 67)
Affinity DataEC50:  31.6nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277261(US10072005, Example 54)
Affinity DataEC50:  31.6nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277266(US10072005, Example 59)
Affinity DataEC50:  39.8nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277269(US10072005, Example 62)
Affinity DataEC50:  39.8nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277286(US10072005, Example 79)
Affinity DataEC50:  39.8nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277221(US10072005, Example 14)
Affinity DataEC50:  50.1nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277292(US10072005, Example 85)
Affinity DataEC50:  50.1nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277271(US10072005, Example 64)
Affinity DataEC50:  63.1nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277288(US10072005, Example 81)
Affinity DataEC50:  63.1nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277287(US10072005, Example 80)
Affinity DataEC50:  79.4nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277249(US10072005, Example 42)
Affinity DataEC50:  100nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277268(US10072005, Example 61)
Affinity DataEC50:  100nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277222(US10072005, Example 15)
Affinity DataEC50:  100nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277208(US10072005, Example 1)
Affinity DataEC50:  100nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277240(US10072005, Example 33)
Affinity DataEC50:  100nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277305(US10072005, Example 98)
Affinity DataEC50:  100nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277308(US10072005, Example 101)
Affinity DataEC50:  100nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277277(US10072005, Example 70)
Affinity DataEC50:  100nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277218(US10072005, Example 11)
Affinity DataEC50:  126nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277251(US10072005, Example 44)
Affinity DataEC50:  126nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277300(US10072005, Example 93)
Affinity DataEC50:  126nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277224(US10072005, Example 17)
Affinity DataEC50:  126nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277304(US10072005, Example 97)
Affinity DataEC50:  126nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277241(US10072005, Example 34)
Affinity DataEC50:  126nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277212(US10072005, Example 5)
Affinity DataEC50:  126nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277210(US10072005, Example 3)
Affinity DataEC50:  158nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM277211(US10072005, Example 4)
Affinity DataEC50:  158nMT: 2°CAssay Description:Following agonist data acquisition, cells were then incubated for a further 30 min at room temperature before either an EC20 concentration (to measur...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2018
Entry Details
US Patent

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