Compile Data Set for Download or QSAR
Report error Found 24 Enz. Inhib. hit(s) with all data for entry = 746
LigandChemical structure of BindingDB Monomer ID 289045BDBM289045(US10093650, Example 22)
Affinity DataIC50: 2nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 289043BDBM289043(US10093650, Example 20 | US10329273, Example 20 | ...)
Affinity DataIC50: 3nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 289021BDBM289021(US10093650, Example 17 | BDBM400246)
Affinity DataIC50: 5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 38176BDBM38176(US10093650, Example 2 | US10329273, Example 2 | US...)
Affinity DataIC50: 5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 289003BDBM289003(US10093650, Example 16 | US10093650, Example 14 | ...)
Affinity DataIC50: 5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 289003BDBM289003(US10093650, Example 16 | US10093650, Example 14 | ...)
Affinity DataIC50: 5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 289026BDBM289026(US10093650, Example 18 | US10329273, Example 18 | ...)
Affinity DataIC50: 8nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 211296BDBM211296(US10093650, Example 11 | US10329273, Example 11 | ...)
Affinity DataIC50: 9nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 289042BDBM289042(US10093650, Example 19 | US10329273, Example 19 | ...)
Affinity DataIC50: 10nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 289044BDBM289044(US10093650, Example 21 | US10329273, Example 21 | ...)
Affinity DataIC50: 10nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 38181BDBM38181(US10093650, Example 4 | US10329273, Example 4 | US...)
Affinity DataIC50: 17nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 38169BDBM38169(US10093650, Example 1 | (S)-3-(5-Oxo-4,5-dihydro-1...)
Affinity DataIC50: 27nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 38204BDBM38204(US10093650, Example 8 | US10329273, Example 8 | US...)
Affinity DataIC50: 30nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 286509BDBM286509(US10093650, Example 12 | US10329273, Example 12 | ...)
Affinity DataIC50: 34nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 289081BDBM289081(US10093650, Example 24 | US11479538, Example 24)
Affinity DataIC50: 36nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 38208BDBM38208(US10093650, Example 10 | US10329273, Example 10 | ...)
Affinity DataIC50: 36nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 289046BDBM289046(US10093650, Example 23 | US10329273, Example 24 | ...)
Affinity DataIC50: 60nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 38191BDBM38191(US10093650, Example 5 | US10329273, Example 5 | US...)
Affinity DataIC50: 71nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 286511BDBM286511(US10093650, Example 13 | US10329273, Example 13 | ...)
Affinity DataIC50: 84nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 38207BDBM38207(US10093650, Example 9 | US10329273, Example 9 | US...)
Affinity DataIC50: 108nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 38192BDBM38192(US10093650, Example 6 | US10329273, Example 6 | US...)
Affinity DataIC50: 137nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 289014BDBM289014(US10093650, Example 15 | US10329273, Example 15 | ...)
Affinity DataIC50: 145nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 38199BDBM38199(US10093650, Example 7 | US10329273, Example 22 | U...)
Affinity DataIC50: 173nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 38179BDBM38179(US10093650, Example 3 | US10329273, Example 3 | US...)
Affinity DataIC50: 340nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/22/2019
Entry Details
US Patent