Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 1162
TargetTGF-beta receptor type-1(Human)
Tiumbio

US Patent
LigandChemical structure of BindingDB Monomer ID 311398BDBM311398(US10155763, Example 6)
Affinity DataIC50: 6.10nMAssay Description:The kinase activity of ALK5 was assessed by measuring radiolabelled phosphate[33P] incorporation into the generic substrate, casein. The kinase domai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Tiumbio

US Patent
LigandChemical structure of BindingDB Monomer ID 311395BDBM311395(US10155763, Example 2)
Affinity DataIC50: 6.60nMAssay Description:The kinase activity of ALK5 was assessed by measuring radiolabelled phosphate[33P] incorporation into the generic substrate, casein. The kinase domai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Tiumbio

US Patent
LigandChemical structure of BindingDB Monomer ID 311399BDBM311399(US10155763, Example 7)
Affinity DataIC50: 10.3nMAssay Description:The kinase activity of ALK5 was assessed by measuring radiolabelled phosphate[33P] incorporation into the generic substrate, casein. The kinase domai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Tiumbio

US Patent
LigandChemical structure of BindingDB Monomer ID 311400BDBM311400(US10155763, Example 9)
Affinity DataIC50: 11.5nMAssay Description:The kinase activity of ALK5 was assessed by measuring radiolabelled phosphate[33P] incorporation into the generic substrate, casein. The kinase domai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Tiumbio

US Patent
LigandChemical structure of BindingDB Monomer ID 311397BDBM311397(US10155763, Example 4)
Affinity DataIC50: 12.1nMAssay Description:The kinase activity of ALK5 was assessed by measuring radiolabelled phosphate[33P] incorporation into the generic substrate, casein. The kinase domai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Tiumbio

US Patent
LigandChemical structure of BindingDB Monomer ID 311396BDBM311396(US10155763, Example 3)
Affinity DataIC50: 31.6nMAssay Description:The kinase activity of ALK5 was assessed by measuring radiolabelled phosphate[33P] incorporation into the generic substrate, casein. The kinase domai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Tiumbio

US Patent
LigandChemical structure of BindingDB Monomer ID 311401BDBM311401(US10155763, Example 15)
Affinity DataIC50: 38.1nMAssay Description:The kinase activity of ALK5 was assessed by measuring radiolabelled phosphate[33P] incorporation into the generic substrate, casein. The kinase domai...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2019
Entry Details
US Patent