Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 1375
TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318948(US10173990, Example 72 | 2-Methyl-2-[[7-(4-nitroph...)
Affinity DataIC50: 12nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318954(US10173990, Example 113 | 2-[[7-(4-Cyanophenyl)ben...)
Affinity DataIC50: 21nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318946(US10173990, Example 66 | 1-[[7-(4-Cyanophenyl)benz...)
Affinity DataIC50: 21.5nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318956(US10173990, Example 116 | (E)-3-[[1-(4-cyanophenyl...)
Affinity DataIC50: 25nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318947(US10173990, Example 68 | 1-[[7-(4-Cyanophenyl)benz...)
Affinity DataIC50: 26.2nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318949(US10173990, Example 78 | 2-Methyl-2-[[7-[4-(triflu...)
Affinity DataIC50: 104nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318950(US10173990, Example 82 | 2-[[7-(4-Chlorophenyl)ben...)
Affinity DataIC50: 106nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318952(US10173990, Example 90 | 2-[[7-(4-Cyano-3-fluoroph...)
Affinity DataIC50: 161nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318944(US10173990, Example 24 | 2-[[7-(4-Cyanophenyl)benz...)
Affinity DataIC50: 170nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318951(US10173990, Example 84 | 2-[[7-(3-Cyanophenyl)benz...)
Affinity DataIC50: 205nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318957(US10173990, Example 117 | 1-[[7-(4-Cyanophenyl)ben...)
Affinity DataIC50: 296nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318955(US10173990, Example 114 | 2-[[7-(4-Cyanophenyl)ben...)
Affinity DataIC50: 474nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318942(US10173990, Example 4 | 2-[(4′-Cyano[1,1R...)
Affinity DataIC50: 790nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318945(US10173990, Example 45 | 2-[[3-(4-Cyanophenyl)quin...)
Affinity DataIC50: 1.58E+3nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318941(US10173990, Example 2 | 2-[(4′-Cyano-(1,1...)
Affinity DataIC50: 2.06E+3nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
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Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318953(US10173990, Example 112 | 1-[[7-(4-Cyanophenyl)-3-...)
Affinity DataIC50: 2.43E+3nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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TargetSolute carrier family 22 member 12(Human)
Nippon Chemiphar

US Patent
LigandPNGBDBM318943(US10173990, Example 15 | 2-[[5-(4-Cyanophenyl)quin...)
Affinity DataIC50: 3.44E+3nMAssay Description:URAT1 stably expressed HEK293 cells (HEK-URAT1) or HEK293 cells transfected with empty vector (HEK-mock) were cultured in DMEM culture medium supplem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2019
Entry Details
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