Compile Data Set for Download or QSAR
Report error Found 234 Enz. Inhib. hit(s) with all data for entry = 1400
LigandChemical structure of BindingDB Monomer ID 320554BDBM320554([4-(Dimethylamino)piperidin-1-yl][5-(1,3-dimethyl-...)
Affinity DataIC50: 3nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320554BDBM320554([4-(Dimethylamino)piperidin-1-yl][5-(1,3-dimethyl-...)
Affinity DataIC50: 3nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320553BDBM320553([5-(1,3-Dimethyl-1H-pyrazol-4-yl)-6-fluoro-7-(morp...)
Affinity DataIC50: 3nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320544BDBM320544(US10174035, Compound 87 | [5-(1,3-Dimethyl-1H-pyra...)
Affinity DataIC50: 3nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320591BDBM320591(US10174035, Compound 134 | [4-(Morpholin-4-yl)pipe...)
Affinity DataIC50: 3nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320544BDBM320544(US10174035, Compound 87 | [5-(1,3-Dimethyl-1H-pyra...)
Affinity DataIC50: 3nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320580BDBM320580(US10174035, Compound 123 | {6-Fluoro-7-(morpholin-...)
Affinity DataIC50: 4nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320551BDBM320551([5-(1,3-Dimethyl-1H-pyrazol-4-yl)-7-(morpholin-4-y...)
Affinity DataIC50: 4nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320551BDBM320551([5-(1,3-Dimethyl-1H-pyrazol-4-yl)-7-(morpholin-4-y...)
Affinity DataIC50: 4nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320541BDBM320541(US10174035, Compound 84 | [5-(1,3-Dimethyl-1H-pyra...)
Affinity DataIC50: 5nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320576BDBM320576(US10174035, Compound 119 | {3-[(2R,6S)-2,6-dimethy...)
Affinity DataIC50: 5nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320570BDBM320570({4-[cis-2,6-Dimethylmorpholin-4-yl]piperidin-1-yl}...)
Affinity DataIC50: 6nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320555BDBM320555([6-Fluoro-5-(1-methyl-1H-pyrazol-4-yl)-7-(morpholi...)
Affinity DataIC50: 6nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320555BDBM320555([6-Fluoro-5-(1-methyl-1H-pyrazol-4-yl)-7-(morpholi...)
Affinity DataIC50: 6nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320570BDBM320570({4-[cis-2,6-Dimethylmorpholin-4-yl]piperidin-1-yl}...)
Affinity DataIC50: 6nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320537BDBM320537(US10174035, Compound 81 | [6-Fluoro-5-(1-methyl-1H...)
Affinity DataIC50: 7nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320529BDBM320529(US10174035, Compound 74 | 4-(1-{[6-(Morpholin-4-yl...)
Affinity DataIC50: 8nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320496BDBM320496([4-(Morpholin-4-yl)piperidin-1-yl][6-(morpholin-4-...)
Affinity DataIC50: 9nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320532BDBM320532(US10174035, Compound 77 | 4-(1-{[5-(1-Methyl-1H-py...)
Affinity DataIC50: 9nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320462BDBM320462(US10174035, Compound 9 | [2-(1,3-Dimethyl-1H-pyraz...)
Affinity DataIC50: 9nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320586BDBM320586(US10174035, Compound 129 | 1-Methyl-4-(1-{[5-(1-me...)
Affinity DataIC50: 10nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320587BDBM320587(US10174035, Compound 130 | 1-Methyl-4-(1-{[2-(1-me...)
Affinity DataIC50: 10nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320461BDBM320461(US10174035, Compound 8 | 2-(4-{[2-(1,3-Dimethyl-1H...)
Affinity DataIC50: 10nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320461BDBM320461(US10174035, Compound 8 | 2-(4-{[2-(1,3-Dimethyl-1H...)
Affinity DataIC50: 10nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320577BDBM320577(US10174035, Compound 120 | [5-(1-Methyl-1H-pyrazol...)
Affinity DataIC50: 10nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320538BDBM320538(US10174035, Compound 82 | 2-(4-{[6-Fluoro-5-(1-met...)
Affinity DataIC50: 11nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320458BDBM320458(US10174035, Compound 5 | {4-[cis-2,6-Dimethylmorph...)
Affinity DataIC50: 11nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320521BDBM320521(US10174035, Compound 67 | 9-Methyl-2-(1-methyl-1H-...)
Affinity DataIC50: 11nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320538BDBM320538(US10174035, Compound 82 | 2-(4-{[6-Fluoro-5-(1-met...)
Affinity DataIC50: 11nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320521BDBM320521(US10174035, Compound 67 | 9-Methyl-2-(1-methyl-1H-...)
Affinity DataIC50: 11nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320458BDBM320458(US10174035, Compound 5 | {4-[cis-2,6-Dimethylmorph...)
Affinity DataIC50: 11nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320519BDBM320519(US10174035, Compound 65 | {4-[cis-2,6-Dimethylmorp...)
Affinity DataIC50: 12nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320471BDBM320471(US10174035, Compound 17 | {2-[1-Methyl-3-(trifluor...)
Affinity DataIC50: 12nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320519BDBM320519(US10174035, Compound 65 | {4-[cis-2,6-Dimethylmorp...)
Affinity DataIC50: 12nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320534BDBM320534(US10174035, Compound 78 | [5-(1-Methyl-1H-pyrazol-...)
Affinity DataIC50: 13nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320473BDBM320473(US10174035, Compound 19 | [4-(Morpholin-4-yl)piper...)
Affinity DataIC50: 13nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320473BDBM320473(US10174035, Compound 19 | [4-(Morpholin-4-yl)piper...)
Affinity DataIC50: 13nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320534BDBM320534(US10174035, Compound 78 | [5-(1-Methyl-1H-pyrazol-...)
Affinity DataIC50: 13nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320512BDBM320512([2-(1-Methyl-1H-pyrazol-4-yl)-6-(morpholin-4-yl)-9...)
Affinity DataIC50: 14nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320495BDBM320495([2-(1,3-Dimethyl-1H-pyrazol-4-yl)-6-(morpholin-4-y...)
Affinity DataIC50: 14nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320512BDBM320512([2-(1-Methyl-1H-pyrazol-4-yl)-6-(morpholin-4-yl)-9...)
Affinity DataIC50: 14nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320495BDBM320495([2-(1,3-Dimethyl-1H-pyrazol-4-yl)-6-(morpholin-4-y...)
Affinity DataIC50: 14nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320456BDBM320456(US10174035, Compound 3 | [2-(1-Methyl-1H-pyrazol-4...)
Affinity DataIC50: 15nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320569BDBM320569({4-[cis-2,6-Dimethylmorpholin-4-yl]piperidin-1-yl}...)
Affinity DataIC50: 15nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320456BDBM320456(US10174035, Compound 3 | [2-(1-Methyl-1H-pyrazol-4...)
Affinity DataIC50: 15nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320490BDBM320490(N-(Cyclohexylmethyl)-2-(1-methyl-1H-pyrazol-4-yl)-...)
Affinity DataIC50: 15nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320468BDBM320468(US10174035, Compound 14 | [4-(2-Hydroxypropan-2-yl...)
Affinity DataIC50: 16nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320468BDBM320468(US10174035, Compound 14 | [4-(2-Hydroxypropan-2-yl...)
Affinity DataIC50: 16nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320572BDBM320572(US10174035, Compound 115 | 5-(1-Methyl-1H-pyrazol-...)
Affinity DataIC50: 16nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 320518BDBM320518(US10174035, Compound 64 | 2-(1-Methyl-1H-pyrazol-4...)
Affinity DataIC50: 17nMAssay Description:The Kinase-Glo luminescent kinase assay kit (from Promega) was used to measure kinase activity. In this assay, amount of ATP remaining in solution fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/16/2019
Entry Details
US Patent

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