Compile Data Set for Download or QSAR
Report error Found 240 Enz. Inhib. hit(s) with all data for entry = 1630
TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333342(US10196396, Compound 153 | (2S,3R,4S)-2-(8-(((1H-b...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333214(US10196396, Compound 9 | (2S,3R,4S)-2-(8-((3-(trif...)
Affinity DataKi: <10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333349(US10196396, Compound 160 | (2S,3R,4S)-2-(8-(((R)-1...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333228(US10196396, Compound 23 | (2S,3R,4S)-2-(8-((furan-...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333305(US10196396, Compound 116 | (2S,3R,4S)-2-(8-morphol...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333294(US10196396, Compound 89 | (2S,3R,4S)-2-(8-((3-phen...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333259(US10196396, Compound 54 | (2S,3R,4S)-2-(8-(2-(3-ch...)
Affinity DataKi: <10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333316(US10196396, Compound 127 | (2S,3R,4S)-2-(8-((3-flu...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333260(US10196396, Compound 55 | (2S,3R,4S)-2-(8-((3,5-di...)
Affinity DataKi: <10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333208(US10196396, Compound 3 | (2S,3R,4S)-2-(8-(piperidi...)
Affinity DataKi: <10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333297(US10196396, Compound 92 | (2S,3R,4S)-2-(8-((3-chlo...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333261(US10196396, Compound 56 | (2S,3R,4S)-2-(8-((2,5-di...)
Affinity DataKi: <10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333221(US10196396, Compound 16 | 3-(((3-((2S,3R,4S)-3,4-d...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333228(US10196396, Compound 23 | (2S,3R,4S)-2-(8-((furan-...)
Affinity DataKi: <10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333265(US10196396, Compound 60 | (2S,3R,4S)-2-(8-((2,4-di...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333227(US10196396, Compound 22 | (2S,3R,4S)-2-(8-((pyridi...)
Affinity DataKi: <10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333359(US10196396, Compound 170 | (2S,3R,4S)-2-(8-((4-flu...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333358(US10196396, Compound 169 | (2S,3R,4S)-2-(8-((2-flu...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333360(US10196396, Compound 171 | Methyl 5-(((3-((2S,3R,4...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333246(US10196396, Compound 41 | (2S,3R,4S)-2-(8-((4-meth...)
Affinity DataKi: <10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333237(US10196396, Compound 32 | (2S,3R,4S)-2-(8-(isopent...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333230(US10196396, Compound 25 | (2S,3R,4S)-2-(8-((3-brom...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333356(US10196396, Compound 167 | 3-chloro-N-(3-((2S,3R,4...)
Affinity DataIC50: 10nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333315(US10196396, Compound 126 | 2-chloro-4-(((3-((2S,3R...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333247(US10196396, Compound 42 | (2S,3R,4S)-2-(8-(morphol...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333318(US10196396, Compound 129 | (2S,3R,4S)-2-(8-((2-phe...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333329(US10196396, Compound 140 | (2S,3R,4S)-2-(8-((3-(tr...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333330(US10196396, Compound 141 | 3-(((3-((2S,3R,4S)-3,4-...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333331(US10196396, Compound 142 | (2S,3R,4S)-2-(8-((pyrim...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333334(US10196396, Compound 145 | (2S,3R,4S)-2-(8-((pyrim...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333325(US10196396, Compound 136 | (2S,3R,4S)-2-(8-((pyrid...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333343(US10196396, Compound 154 | (2S,3R,4S)-2-(8-((2-(pi...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333345(US10196396, Compound 156 | (2S,3R,4S)-2-(8-((2-(di...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333344(US10196396, Compound 155 | (2S,3R,4S)-2-(8-((3-chl...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333347(US10196396, Compound 158 | 3-chloro-N-(3-((2S,3R,4...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333348(US10196396, Compound 159 | (2S,3R,4S)-2-(8-((3-chl...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333335(US10196396, Compound 146 | (2S,3R,4S)-2-(8-((3-chl...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333261(US10196396, Compound 56 | (2S,3R,4S)-2-(8-((2,5-di...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333337(US10196396, Compound 148 | (2S,3R,4S)-2-(8-((thiaz...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333336(US10196396, Compound 147 | (2S,3R,4S)-2-(8-((thiaz...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333339(US10196396, Compound 150 | (2S,3R,4S)-2-(8-((2-mor...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333338(US10196396, Compound 149 | (2S,3R,4S)-2-(8-((3-bro...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333341(US10196396, Compound 152 | (2S,3R,4S)-2-(8-((2-(3-...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333340(US10196396, Compound 151 | (2S,3R,4S)-2-(8-((1-(3-...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333263(US10196396, Compound 58 | (2S,3R,4S)-2-(8-((2,3-di...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333262(US10196396, Compound 57 | (2S,3R,4S)-2-(8-((thioph...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333264(US10196396, Compound 59 | (2S,3R,4S)-2-(8-((3,4-di...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333350(US10196396, Compound 161 | (2S,3R,4S)-2-(8-(((S)-1...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333353(US10196396, Compound 164 | (2S,3R,4S)-2-(8-((4-chl...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
Handok

US Patent
LigandPNGBDBM333352(US10196396, Compound 163 | (2S,3R,4S)-2-(8-((2-chl...)
Affinity DataIC50: 55nMAssay Description:HEK-293 cell membrane homogenates (32 μg protein), in which A3 adenosine receptors were expressed, are incubated for 120 min at 22° C. with 0.15...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2019
Entry Details
US Patent

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