Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 2179
TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357011BDBM357011(5-Amino-1-(3-fluoro-2-methylphenyl)-N-(5-(trifluor...)
Affinity DataIC50: 200nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357010BDBM357010(5-Amino-1-(2-hydroxyphenyl)-N-(5-(trifluoromethyl)...)
Affinity DataIC50: 300nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 356996BDBM356996(5-Amino-N-(4-chloro-2-fluoro-phenyl)-1-(o-tolyl)-1...)
Affinity DataIC50: 300nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357006BDBM357006(5-Amino-3-ethyl-1-(3-fluoro-2-methylphenyl)-N-[5-t...)
Affinity DataIC50: 300nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357002BDBM357002(5-Amino-3-ethyl-1-(2-methoxyphenyl)-N-(5-(trifluor...)
Affinity DataIC50: 400nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357007BDBM357007(5-Amino-1-(2-fluorophenyl)-3-methyl-N-(5-(trifluor...)
Affinity DataIC50: 400nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 356998BDBM356998(5-Amino-1-(3-fluoro-2-methylphenyl)-N-(5-(trifluor...)
Affinity DataIC50: 500nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357004BDBM357004(5-Amino-N-(5-chloro-2-pyridyl)-1-(3-fluoro-2-methy...)
Affinity DataIC50: 600nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 356995BDBM356995(5-Amino-N-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-...)
Affinity DataIC50: 700nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357003BDBM357003(5-Amino-1-(2-(2-methoxyethoxy)phenyl)-3-methyl-N-(...)
Affinity DataIC50: 700nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 356997BDBM356997(5-Amino-N-(2-fluoro-4-(trifluoromethyl)phenyl)-1-(...)
Affinity DataIC50: 700nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357008BDBM357008(5-Amino-N-(5-chloropyridin-2-yl)-1-(2-(pyridin-3-y...)
Affinity DataIC50: 700nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357001BDBM357001(5-Amino-N-(5-chloropyridin-2-yl)-1-(3-fluoro-2-met...)
Affinity DataIC50: 800nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 356999BDBM356999((5-Amino-1-(3-fluoro-2-methylphenyl)-1H-pyrazol-4-...)
Affinity DataIC50: 800nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357000BDBM357000((5-Amino-1-(2-methoxyphenyl)-1H-pyrazol-4-yl)(5-ch...)
Affinity DataIC50: 900nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357009BDBM357009(5-Amino-N-(5-chloropyridin-2-yl)-1-(2-(2-methoxypy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357005BDBM357005(5-Amino-1-(2-ethylphenyl)-N-(5-(2,2,2-trifluoroeth...)
Affinity DataIC50: 1.00E+3nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 9 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357012BDBM357012(5-Amino-N-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-...)
Affinity DataIC50: 1.90E+3nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357006BDBM357006(5-Amino-3-ethyl-1-(3-fluoro-2-methylphenyl)-N-[5-t...)
Affinity DataIC50: 1.00E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357008BDBM357008(5-Amino-N-(5-chloropyridin-2-yl)-1-(2-(pyridin-3-y...)
Affinity DataIC50: 1.70E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 356995BDBM356995(5-Amino-N-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-...)
Affinity DataIC50: 2.10E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357000BDBM357000((5-Amino-1-(2-methoxyphenyl)-1H-pyrazol-4-yl)(5-ch...)
Affinity DataIC50: 2.80E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357010BDBM357010(5-Amino-1-(2-hydroxyphenyl)-N-(5-(trifluoromethyl)...)
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357009BDBM357009(5-Amino-N-(5-chloropyridin-2-yl)-1-(2-(2-methoxypy...)
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357012BDBM357012(5-Amino-N-(4-chlorophenyl)-1-(2-methoxyphenyl)-1H-...)
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 356996BDBM356996(5-Amino-N-(4-chloro-2-fluoro-phenyl)-1-(o-tolyl)-1...)
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357005BDBM357005(5-Amino-1-(2-ethylphenyl)-N-(5-(2,2,2-trifluoroeth...)
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357007BDBM357007(5-Amino-1-(2-fluorophenyl)-3-methyl-N-(5-(trifluor...)
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357002BDBM357002(5-Amino-3-ethyl-1-(2-methoxyphenyl)-N-(5-(trifluor...)
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357001BDBM357001(5-Amino-N-(5-chloropyridin-2-yl)-1-(3-fluoro-2-met...)
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357004BDBM357004(5-Amino-N-(5-chloro-2-pyridyl)-1-(3-fluoro-2-methy...)
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 357003BDBM357003(5-Amino-1-(2-(2-methoxyethoxy)phenyl)-3-methyl-N-(...)
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 356998BDBM356998(5-Amino-1-(3-fluoro-2-methylphenyl)-N-(5-(trifluor...)
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 356997BDBM356997(5-Amino-N-(2-fluoro-4-(trifluoromethyl)phenyl)-1-(...)
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent

TargetSodium channel protein type 5 subunit alpha(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 356999BDBM356999((5-Amino-1-(3-fluoro-2-methylphenyl)-1H-pyrazol-4-...)
Affinity DataIC50: 3.30E+4nMAssay Description:Cell LinesStable cell lines expressing the full-length protein of the voltage-gated sodium channels Nav1.7 or Nav1.5, with or without one beta-1, bet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/20/2019
Entry Details
US Patent