Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 3117
TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391797BDBM391797(US10300067, Example 49 | 6-((7-(3-Chloro-4-cyanoph...)
Affinity DataIC50: 2nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391776BDBM391776(US10300067, Example 28 | 6-((7-(4-Cyano-3-(trifluo...)
Affinity DataIC50: 20nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391759BDBM391759(US10300067, Example 11 | 6-((7-(4-Cyano-3-(trifluo...)
Affinity DataIC50: 30nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391789BDBM391789(US10300067, Example 42 | 4-(4-((5-(4-(2-Hydroxypro...)
Affinity DataIC50: 34nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391792BDBM391792(US10300067, Example 44 | 2-Bromo-4-(4-((5-(2-hydro...)
Affinity DataIC50: 50nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391802BDBM391802(US10300067, Example 53 | 2-Chloro-4-(4-((5-(2-meth...)
Affinity DataIC50: 55nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391774BDBM391774(US10300067, Example 26 | 2-((7-(4-Cyano-3-(trifluo...)
Affinity DataIC50: 60nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391779BDBM391779(US10300067, Example 32 | 6-((7-(4-Cyano-3-(trifluo...)
Affinity DataIC50: 60nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391772BDBM391772(US10300067, Example 24 | 6-((7-(4-Cyano-3-(trifluo...)
Affinity DataIC50: 70nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391752BDBM391752(US10300067, Example 6 | 2-Chloro-4-(4-((6-(2-hydro...)
Affinity DataIC50: 70nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391795BDBM391795(US10300067, Example 47 | 4-(4-((4-Fluoro-5-(2-hydr...)
Affinity DataIC50: 70nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391730BDBM391730(US10300067, Example 1 | 4-(4-((1,2,4-Thiadiazol-5-...)
Affinity DataIC50: 80nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391775BDBM391775(US10300067, Example 27 | 6-((7-(4-Cyano-3-(trifluo...)
Affinity DataIC50: 90nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391758BDBM391758(US10300067, Example 10 | 4-(4-((6-(2-Hydroxypropan...)
Affinity DataIC50: 90nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391768BDBM391768(US10300067, Example 20 | 4-(4-((5-((1,4-Oxazepan-4...)
Affinity DataIC50: 100nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391761BDBM391761(US10300067, Example 13 | 4-(4-((6-Isopropoxypyridi...)
Affinity DataIC50: 110nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391763BDBM391763(US10300067, Example 15 | 4-(4-((6-(2-(1H-1,2,3-Tri...)
Affinity DataIC50: 130nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391767BDBM391767(US10300067, Example 19 | 6-((7-(4-Cyano-3-(trifluo...)
Affinity DataIC50: 130nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391800BDBM391800(US10300067, Example 52 | 4-(4-((5-Chloro-6-(2-meth...)
Affinity DataIC50: 150nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391753BDBM391753(US10300067, Example 7 | 4-(4-((5-(2-Hydroxypropan-...)
Affinity DataIC50: 160nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391760BDBM391760(US10300067, Example 12 | 4-(4-((5-(1-Hydroxycyclop...)
Affinity DataIC50: 170nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391765BDBM391765(US10300067, Example 17 | 4-(4-((5-(2-Methyl-2-(1H-...)
Affinity DataIC50: 170nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391784BDBM391784(US10300067, Example 37 | (R)—N-(1-(1,3,4-Oxad...)
Affinity DataIC50: 170nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391783BDBM391783(US10300067, Example 36 | 6-((7-(4-Cano-3-(trifluor...)
Affinity DataIC50: 170nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391751BDBM391751(US10300067, Example 5 | 4-(4-((6-Fluoro-5-(2-hydro...)
Affinity DataIC50: 190nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391782BDBM391782(US10300067, Example 35 | 5-((7-(4-Cano-3-(trifluor...)
Affinity DataIC50: 190nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391777BDBM391777(US10300067, Example 29 | 6-((7-(3-Chloro-4-cyanoph...)
Affinity DataIC50: 200nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391764BDBM391764(US10300067, Example 16 | 4-(4-((6-(2-Methyl-2-(1H-...)
Affinity DataIC50: 210nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391755BDBM391755(US10300067, Example 9 | 2-Chloro-4-(4-((5-(2-hydro...)
Affinity DataIC50: 250nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391754BDBM391754(US10300067, Example 8 | 4-(4-((5-(2-Hydroxypropan-...)
Affinity DataIC50: 250nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391794BDBM391794(US10300067, Example 46 | 2-Chloro-4-(4-((6-fluoro-...)
Affinity DataIC50: 250nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391787BDBM391787(US10300067, Example 40 | (R)-6-((7-(4-Cyano-3-(tri...)
Affinity DataIC50: 260nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391762BDBM391762(US10300067, Example 14 | 4-(4-((4-(2-(1-Methyl-1H-...)
Affinity DataIC50: 300nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391780BDBM391780(US10300067, Example 33 | 5-((7-(4-Cyano-3-(trifluo...)
Affinity DataIC50: 310nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391798BDBM391798(US10300067, Example 50 | 4-(4-((5-Fluoro-6-(2-meth...)
Affinity DataIC50: 320nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391766BDBM391766(US10300067, Example 18 | 4-(4-((4-(3-(4-(Methylsul...)
Affinity DataIC50: 360nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391770BDBM391770(US10300067, Example 22 | 2-(6-((7-(4-Cyano-3-(trif...)
Affinity DataIC50: 370nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391748BDBM391748(US10300067, Example 2 | 4-(4-((4-Isopropoxyphenyl)...)
Affinity DataIC50: 370nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391769BDBM391769(US10300067, Example 21 | 2,2,2-Trifluoroethyl (6-(...)
Affinity DataIC50: 380nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391778BDBM391778(US10300067, Example 31 | 2-((7-(4-Cyano-3-(trifluo...)
Affinity DataIC50: 390nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391796BDBM391796(US10300067, Example 48 | 5-((7-(4-Cyano-3-(trifluo...)
Affinity DataIC50: 490nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391749BDBM391749(US10300067, Example 3 | 4-(4-((4-Methoxyphenyl)ami...)
Affinity DataIC50: 530nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391785BDBM391785(US10300067, Example 38 | (R)—N-(1-(1,3,4-Oxad...)
Affinity DataIC50: 560nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391750BDBM391750(US10300067, Example 4 | 4-(4-((1,1′-Biphenyl...)
Affinity DataIC50: 620nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391781BDBM391781(US10300067, Example 34 | 2-((7-(4-Cyano-3-(trifluo...)
Affinity DataIC50: 700nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391791BDBM391791(US10300067, Example 43 | 4-(4-((5-(4-(2-Hydroxypro...)
Affinity DataIC50: 790nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391771BDBM391771(US10300067, Example 23 | N-(6-((7-(4-Cano-3-(trifl...)
Affinity DataIC50: 800nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391803BDBM391803(US10300067, Example 56 | 2-Chloro-4-(4-((6-fluoro-...)
Affinity DataIC50: 840nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391793BDBM391793(US10300067, Example 45 | 2-Chloro-4-(4-((4-fluoro-...)
Affinity DataIC50: 940nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

TargetAndrogen receptor(Human)
Taiho Pharmaceutical

US Patent
LigandChemical structure of BindingDB Monomer ID 391799BDBM391799(US10300067, Example 51 | 4-(4-((5-Fluoro-6-(2-meth...)
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity for AR was evaluated according to the following method. COS-7 cells (ATCC) were transfected with pMMTV-luc vector (reporter plasm...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/25/2020
Entry Details
US Patent

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