Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 8821
TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420962BDBM420962(US10479798, Compound 21)
Affinity DataIC50: 2nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoPDBSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 50198186BDBM50198186(CHEMBL3944427 | US10479798, Compound 19)
Affinity DataIC50: 2nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 50003020BDBM50003020(MK-3102 | OMARIGLIPTIN | US10155775, Omarigliptin ...)
Affinity DataIC50: 2nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420415BDBM420415(US10479798, Compound 12)
Affinity DataIC50: 4nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 50198175BDBM50198175(CHEMBL3932825 | US10479798, Compound 17)
Affinity DataIC50: 6nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420402BDBM420402(US10479798, Compound 9)
Affinity DataIC50: 9.17nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420956BDBM420956(US10479798, Compound 16)
Affinity DataIC50: 11nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 11162BDBM11162(Triazolopiperazine Analogue 1 | (3R)-3-amino-1-[3-...)
Affinity DataIC50: 14nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 50198180BDBM50198180(CHEMBL3928073 | US10479798, Compound 5)
Affinity DataIC50: 15nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420408BDBM420408(US10479798, Compound 10)
Affinity DataIC50: 18nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 50198178BDBM50198178(CHEMBL3901191 | US10479798, Compound 6)
Affinity DataIC50: 20nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 50198184BDBM50198184(CHEMBL3942843 | US10479798, Compound 20)
Affinity DataIC50: 30nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420966BDBM420966(US10479798, Compound 25)
Affinity DataIC50: 33nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 50198185BDBM50198185(CHEMBL3979508 | US10479798, Compound 7)
Affinity DataIC50: 39nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420971BDBM420971(US10479798, Compound 30)
Affinity DataIC50: 55nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420969BDBM420969(US10479798, Compound 28)
Affinity DataIC50: 56nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420958BDBM420958(US10479798, Compound 18)
Affinity DataIC50: 70nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420477BDBM420477(US10479798, Compound 14)
Affinity DataIC50: 74nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420965BDBM420965(US10479798, Compound 24)
Affinity DataIC50: 78nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420854BDBM420854(US10479798, Compound 15)
Affinity DataIC50: 110nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 50198164BDBM50198164(CHEMBL3959577 | US10479798, Compound 3)
Affinity DataIC50: 154nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420453BDBM420453(US10479798, Compound 13)
Affinity DataIC50: 169nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420412BDBM420412(US10479798, Compound 11)
Affinity DataIC50: 205nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420328BDBM420328(US10479798, Compound 2)
Affinity DataIC50: 207nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420400BDBM420400(US10479798, Compound 8)
Affinity DataIC50: 216nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420970BDBM420970(US10479798, Compound 29)
Affinity DataIC50: 254nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420338BDBM420338(US10479798, Compound 4)
Affinity DataIC50: 283nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420967BDBM420967(US10479798, Compound 26)
Affinity DataIC50: 338nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420963BDBM420963(US10479798, Compound 22)
Affinity DataIC50: 564nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420968BDBM420968(US10479798, Compound 27)
Affinity DataIC50: 678nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420964BDBM420964(US10479798, Compound 23)
Affinity DataIC50: 800nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent

TargetDipeptidyl peptidase 4(Human)
East China University of Science and Technology

US Patent
LigandChemical structure of BindingDB Monomer ID 420322BDBM420322(US10479798, Compound 1)
Affinity DataIC50: 3.32E+3nMAssay Description:Screening Method:Name of method: Activity Evaluation of DPP4, Fluorescence.Instrument: Microplate reader, Envision (PerkinElmer, USA).Material: human...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
9/25/2020
Entry Details
US Patent