Compile Data Set for Download or QSAR
Report error Found 120 Enz. Inhib. hit(s) with all data for entry = 8832
TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421947BDBM421947(US10494376, Example 55)
Affinity DataIC50: 16nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 422000BDBM422000(US10494376, Example 108)
Affinity DataIC50: 17nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421943BDBM421943(US10494376, Example 50)
Affinity DataIC50: 19nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421942BDBM421942(US10494376, Example 49)
Affinity DataIC50: 38nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421997BDBM421997(US10494376, Example 105)
Affinity DataIC50: 38nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421920BDBM421920(US10494376, Example 27)
Affinity DataIC50: 44nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421973BDBM421973(US10494376, Example 81)
Affinity DataIC50: 51nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421919BDBM421919(US10494376, Example 26)
Affinity DataIC50: 53nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421979BDBM421979(US10494376, Example 87)
Affinity DataIC50: 57nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421944BDBM421944(US10494376, Example 51)
Affinity DataIC50: 61nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421975BDBM421975(US10494376, Example 83)
Affinity DataIC50: 65nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421995BDBM421995(US10494376, Example 103)
Affinity DataIC50: 65nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421992BDBM421992(US10494376, Example 100)
Affinity DataIC50: 66nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421994BDBM421994(US10494376, Example 102)
Affinity DataIC50: 68nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421914BDBM421914(US10494376, Example 21)
Affinity DataIC50: 70nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 422011BDBM422011(US10494376, Example 124)
Affinity DataIC50: 70nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421954BDBM421954(US10494376, Example 62)
Affinity DataIC50: 102nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421993BDBM421993(US10494376, Example 101)
Affinity DataIC50: 104nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421953BDBM421953(US10494376, Example 61)
Affinity DataIC50: 104nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421930BDBM421930(US10494376, Example 37)
Affinity DataIC50: 105nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421974BDBM421974(US10494376, Example 82)
Affinity DataIC50: 106nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421962BDBM421962(US10494376, Example 70)
Affinity DataIC50: 121nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421983BDBM421983(US10494376, Example 91)
Affinity DataIC50: 123nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421976BDBM421976(US10494376, Example 84)
Affinity DataIC50: 124nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421991BDBM421991(US10494376, Example 99)
Affinity DataIC50: 127nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421923BDBM421923(US10494376, Example 30)
Affinity DataIC50: 139nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421996BDBM421996(US10494376, Example 104)
Affinity DataIC50: 147nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421929BDBM421929(US10494376, Example 36)
Affinity DataIC50: 148nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421928BDBM421928(US10494376, Example 35)
Affinity DataIC50: 152nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421972BDBM421972(US10494376, Example 80)
Affinity DataIC50: 161nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421971BDBM421971(US10494376, Example 79)
Affinity DataIC50: 168nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421921BDBM421921(US10494376, Example 28)
Affinity DataIC50: 180nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421980BDBM421980(US10494376, Example 88)
Affinity DataIC50: 187nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421941BDBM421941(US10494376, Example 48)
Affinity DataIC50: 192nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421981BDBM421981(US10494376, Example 89)
Affinity DataIC50: 203nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421924BDBM421924(US10494376, Example 31)
Affinity DataIC50: 204nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421935BDBM421935(US10494376, Example 42)
Affinity DataIC50: 212nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421998BDBM421998(US10494376, Example 106)
Affinity DataIC50: 212nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421990BDBM421990(US10494376, Example 98)
Affinity DataIC50: 230nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421939BDBM421939(US10494376, Example 46)
Affinity DataIC50: 230nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 422012BDBM422012(US10494376, Example 125)
Affinity DataIC50: 232nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421955BDBM421955(US10494376, Example 63)
Affinity DataIC50: 245nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421956BDBM421956(US10494376, Example 64)
Affinity DataIC50: 261nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421968BDBM421968(US10494376, Example 76)
Affinity DataIC50: 262nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421977BDBM421977(US10494376, Example 85)
Affinity DataIC50: 279nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421926BDBM421926(US10494376, Example 33)
Affinity DataIC50: 305nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421959BDBM421959(US10494376, Example 67)
Affinity DataIC50: 307nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421984BDBM421984(US10494376, Example 92)
Affinity DataIC50: 310nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421958BDBM421958(US10494376, Example 66)
Affinity DataIC50: 329nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

TargetProtein arginine N-methyltransferase 5(Human)
Ctxt

US Patent
LigandChemical structure of BindingDB Monomer ID 421966BDBM421966(US10494376, Example 74)
Affinity DataIC50: 338nMAssay Description:Compounds of the invention may be tested for in vitro activity in the following assay: A histone H4 derived peptide is used as substrate (amino acid ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/2/2020
Entry Details
US Patent

Displayed 1 to 50 (of 120 total ) | Next | Last >>
Jump to: