Compile Data Set for Download or QSAR
Report error Found 167 Enz. Inhib. hit(s) with all data for entry = 8864
TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425103BDBM425103(US10519118, Example 178 | N-((S)-5-((1R,2S)-2-(4- ...)
Affinity DataIC50: 800nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425069BDBM425069(US10519118, Example 147 | N-((S)-4-((1R,2S)-2-(4- ...)
Affinity DataIC50: 1.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424965BDBM424965(US10519118, Example 33 | 4-fluoro-1-((S)-5-((1R,2S...)
Affinity DataIC50: 2.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425104BDBM425104(US10519118, Example 180 | N-((S)-5-((1R,2S)-2-(4- ...)
Affinity DataIC50: 2.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425055BDBM425055(US10519118, Example 128 | N-[(2S)-5-[[(1R,2S)-2-(4...)
Affinity DataIC50: 2.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425102BDBM425102(US10519118, Example 177 | N-((S)-5-((1R,2S)-2-(4- ...)
Affinity DataIC50: 2.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424951BDBM424951(US10519118, Example 19 | N-((S)-4-((1R,2S)-2-(4- m...)
Affinity DataIC50: 3.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425077BDBM425077(US10519118, Example 152 | N-((S)-4-((1R,2S)-2-(4- ...)
Affinity DataIC50: 3.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424966BDBM424966(US10519118, Example 35 | N-[(2S)-1-(3-cyanoazetidi...)
Affinity DataIC50: 3.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424977BDBM424977(US10519118, Example 49 | N-[(2S)-5-[[(1R,2S)-2-(4-...)
Affinity DataIC50: 3.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425101BDBM425101(US10519118, Example 176 | N-((S)-1-(azetidin-1-yl)...)
Affinity DataIC50: 3.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425084BDBM425084(US10519118, Example 159 | N-((S)-4-((1R,2S)-2-(4- ...)
Affinity DataIC50: 3.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425099BDBM425099(US10519118, Example 174 | 4-cyano-N-((S)-5-((1R,2S...)
Affinity DataIC50: 3.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425005BDBM425005(US10519118, Example 75 | 4-Cyano-N-[(2S)-1-(4-ethy...)
Affinity DataIC50: 4.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425020BDBM425020(US10519118, Example 92 | 4-Cyano-N-[(2S)-5-[[(1R,2...)
Affinity DataIC50: 4.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425111BDBM425111(US10519118, Example 187 | 4'-fluoro-N-((S)-4-((1R,...)
Affinity DataIC50: 4.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425105BDBM425105(US10519118, Example 181 | N-((S)-5-((1R,2S)-2-(4- ...)
Affinity DataIC50: 4.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425085BDBM425085(US10519118, Example 160 | N-((S)-4-((1R,2S)-2-(4- ...)
Affinity DataIC50: 4.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424980BDBM424980(US10519118, Example 51 | N-[(2S)-5-[[(1R,2S)-2-(4-...)
Affinity DataIC50: 4.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424962BDBM424962(US10519118, Example 30 | 1-((S)-2-(4-cyanobenzamid...)
Affinity DataIC50: 4.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425096BDBM425096(US10519118, Example 171 | N-((S)-5-((1R,2S)-2-(4- ...)
Affinity DataIC50: 4.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424952BDBM424952(US10519118, Example 20 | N-((S)-4-((1R,2S)-2-(4- f...)
Affinity DataIC50: 5.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424954BDBM424954(US10519118, Example 23 | N-[(2S)-5-[[(1R,2S)-2-(4-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424935BDBM424935(N-((S)-4-((1R,2S)-2-(4- fluorophenyl)cyclopropylam...)
Affinity DataIC50: 5.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425017BDBM425017(US10519118, Example 89 | N-((S)-1-((3S,5R)-3,5-dim...)
Affinity DataIC50: 5.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425039BDBM425039(US10519118, Example 108 | N-[(2S)-5-[[(1R,2S)-2-(4...)
Affinity DataIC50: 5.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425038BDBM425038(US10519118, Example 107 | N-[(2S)-1-[4-(2-Cyanoace...)
Affinity DataIC50: 5.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425071BDBM425071(US10519118, Example 148 | 4-(2,5-dimethyl-1H-pyrro...)
Affinity DataIC50: 5.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425029BDBM425029(US10519118, Example 97 | N-[(2S)-5-[[(1R,2S)-2-(4-...)
Affinity DataIC50: 5.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425097BDBM425097(US10519118, Example 172 | N-((S)-5-((1R,2S)-2-(4- ...)
Affinity DataIC50: 5.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424939BDBM424939(N-((S)-4-((1R,2S)-2-(4- fluorophenyl)cyclopropylam...)
Affinity DataIC50: 5.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424938BDBM424938(4'-fluoro-N-((S)-4-((1R,2S)-2-(4- fluorophenyl)cyc...)
Affinity DataIC50: 5.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425098BDBM425098(US10519118, Example 173 | N-((S)-5-((1R,2S)-2-(4- ...)
Affinity DataIC50: 5.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425018BDBM425018(US10519118, Example 90 | N-[(2S)-5-[[(1R,2S)-2-(4-...)
Affinity DataIC50: 6.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425051BDBM425051(US10519118, Example 123 | N-[(2S)-1-[1,4-Diazabicy...)
Affinity DataIC50: 6.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425087BDBM425087(US10519118, Example 162 | N-((S)-5-((1R,2S)-2-(4- ...)
Affinity DataIC50: 6.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424945BDBM424945(US10519118, Example 13 | N-((S)-4-((1R,2S)-2-(4- f...)
Affinity DataIC50: 6.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425063BDBM425063(US10519118, Example 141 | N-((S)-6-((1R,2S)-2-(4- ...)
Affinity DataIC50: 6.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424940BDBM424940(2-(biphenyl-4-yl)-N-((S)-4-((1R,2S)-2-(4- fluoroph...)
Affinity DataIC50: 6.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425016BDBM425016(US10519118, Example 86 | N-[(2S)-5-[[(1R,2S)-2-(4-...)
Affinity DataIC50: 7.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425068BDBM425068(US10519118, Example 146 | US10519118, Example 149 ...)
Affinity DataIC50: 7.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425048BDBM425048(US10519118, Example 120 | N-[(2S)-5-[[(1R,2S)-2-(4...)
Affinity DataIC50: 7.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424992BDBM424992(US10519118, Example 61 | 1-((S)-2-(4-(1H-1,2,3-tri...)
Affinity DataIC50: 7.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425044BDBM425044(US10519118, Example 115 | N-[(2S)-5-[[(1R,2S)-2-(4...)
Affinity DataIC50: 7.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424968BDBM424968(US10519118, Example 38 | N-[(2S)-5-[[(1R,2S)-2-(4-...)
Affinity DataIC50: 8.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 424964BDBM424964(US10519118, Example 32 | 4-cyano-N-[(2S)-5-[[(1R,2...)
Affinity DataIC50: 8.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425052BDBM425052(US10519118, Example 124 | N-[(2S)-5-[[(1R,2S)-2-(4...)
Affinity DataIC50: 8.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425015BDBM425015(US10519118, Example 85 | N-[(2S)-1-(4-Ethylpiperaz...)
Affinity DataIC50: 8.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425028BDBM425028(US10519118, Example 96 | 4-(Dimethylsulfamoyl)-N-[...)
Affinity DataIC50: 8.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Imago Biosciences

US Patent
LigandChemical structure of BindingDB Monomer ID 425110BDBM425110(US10519118, Example 186 | N-((S)-4-((1R,2S)-2-(4- ...)
Affinity DataIC50: 9.00E+3nMAssay Description:Briefly, bulk histones, histone peptides or nucleosomes are incubated with purified human recombinant KDM1A, in the histone demethylase activity (HDM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/19/2020
Entry Details
US Patent

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