Compile Data Set for Download or QSAR
Report error Found 308 Enz. Inhib. hit(s) with all data for entry = 8964
TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432135BDBM432135(US10577360, Example 2 | N-(1-Benzylpiperidin-4-yl)...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432269BDBM432269(US10577360, Example 132 | N-[6-(4-Methoxyphenyl)py...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432134BDBM432134(US10577360, Example 1 | N-(1-Benzylpiperidin-4-yl)...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432198BDBM432198(US10577360, Example 62 | N-{3-[Benzyl(methyl)amino...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432145BDBM432145(US10577360, Example 11 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432142BDBM432142(US10577360, Example 8 | N-[1-(4-Fluorophenyl)-1H-p...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432143BDBM432143(US10577360, Example 9 | N-[1-(4-Fluorophenyl)-1H-p...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432273BDBM432273(N-(1-benzylpiperidin-4-yl)-N-(1-phenyl-1H-1,2,3-tr...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432139BDBM432139(US10577360, Example 6 | N-(1-Benzylpiperidin-4-yl)...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432272BDBM432272(US10577360, Example 135 | N-(1-benzylpiperidin-4-y...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432137BDBM432137(US10577360, Example 4 | N-(1-Benzylpiperidin-4-yl)...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432273BDBM432273(N-(1-benzylpiperidin-4-yl)-N-(1-phenyl-1H-1,2,3-tr...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432138BDBM432138(US10577360, Example 5 | N-(1-Benzylpiperidin-4-yl)...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432152BDBM432152(US10577360, Example 18 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432254BDBM432254(US10577360, Example 117 | N-(1-Benzylpiperidin-4-y...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432153BDBM432153(US10577360, Example 19 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432150BDBM432150(US10577360, Example 16 | N-(1-Phenethylpiperidin-4...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432219BDBM432219(US10577360, Example 82 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432151BDBM432151(US10577360, Example 17 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432187BDBM432187(US10577360, Example 51 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432220BDBM432220(US10577360, Example 83 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432253BDBM432253(US10577360, Example 116 | N-(1-Benzylpiperidin-4-y...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432250BDBM432250(US10577360, Example 113 | N-{1-[3-(5-Methyl-1,3,4-...)
Affinity DataKi: <100nMAssay Description:Human α2δ-1 enriched membranes (2.5 μg) were incubated with 15 nM of radiolabeled [3H]-Gabapentin in assay buffer containing Hepes-KOH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432148BDBM432148(US10577360, Example 14 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432217BDBM432217(US10577360, Example 80 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432149BDBM432149(US10577360, Example 15 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432185BDBM432185(US10577360, Example 49 | N-(1-phenethylpiperidin-4...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432146BDBM432146(US10577360, Example 12 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432215BDBM432215(US10577360, Example 78 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432248BDBM432248(US10577360, Example 111 | 3-Hydroxy-N-[1-(3-methox...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432147BDBM432147(US10577360, Example 13 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432216BDBM432216(US10577360, Example 79 | N-(1-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432197BDBM432197(US10577360, Example 61 | N-{2-[Benzyl(methyl)amino...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432194BDBM432194(US10577360, Example 58 | N-(1-Isobutylpiperidin-4-...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432290BDBM432290(US10577360, Example 154 | N-{(1s,4s)-4-[Benzyl(met...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432192BDBM432192(US10577360, Example 56 | N-[3-(Benzylamino)propyl]...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432258BDBM432258(US10577360, Example 121 | N-[1-(3-Methoxyphenyl)-1...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432193BDBM432193(US10577360, Example 57 | N-[2-(Methylamino)ethyl]-...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432288BDBM432288(US10577360, Example 152 | N-{(1s,4s)-4-[Benzyl(met...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432190BDBM432190(US10577360, Example 54 | N-(2-Benzylpiperidin-4-yl...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432256BDBM432256(US10577360, Example 119 | N-(1-Benzylpiperidin-4-y...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432289BDBM432289(US10577360, Example 153 | N-{(1r,4r)-4-[Benzyl(met...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432191BDBM432191(US10577360, Example 55 | N-[2-(Benzylamino)ethyl]-...)
Affinity DataKi: <100nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432205BDBM432205(US10577360, Example 68 | N-[2-(Ethylamino)ethyl]-N...)
Affinity DataKi:  300nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432206BDBM432206(US10577360, Example 69 | N-{2-[Benzyl(methyl)amino...)
Affinity DataKi:  300nMAssay Description:Human α2δ-1 enriched membranes (2.5 μg) were incubated with 15 nM of radiolabeled [3H]-Gabapentin in assay buffer containing Hepes-KOH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432136BDBM432136(US10577360, Example 3 | N-(1-Benzylpiperidin-4-yl)...)
Affinity DataKi:  300nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432203BDBM432203(US10577360, Example 66 | N-{2-[Methyl(pyridin-4-yl...)
Affinity DataKi:  300nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432266BDBM432266(US10577360, Example 129 | N-[6-(4-Fluorophenyl)pyr...)
Affinity DataKi:  300nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetVoltage-dependent calcium channel subunit alpha-2/delta-1(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432267BDBM432267(US10577360, Example 130 | N-{6-[3-(5-Methyl-1,3,4-...)
Affinity DataKi:  300nMAssay Description:Human α2δ-1 enriched membranes (2.5 μg) were incubated with 15 nM of radiolabeled [3H]-Gabapentin in assay buffer containing Hepes-KOH...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Esteve Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 432265BDBM432265(US10577360, Example 128 | N-{4-[Benzyl(methyl)amin...)
Affinity DataKi:  300nMAssay Description:To investigate binding properties of test compounds to human μ-opioid receptor, transfected CHO-K1 cell membranes and [3H]-DAMGO (Perkin Elmer, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/20/2020
Entry Details
US Patent

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