Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 9042
TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 286100BDBM286100(US9517228, Example 1 (4'S) | US9987253, Example 1 ...)
Affinity DataIC50: 100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2020
Entry Details
US Patent

TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 397087BDBM397087(US9987253, Example 2 | US10617673, Example 2 | US1...)
Affinity DataIC50: 100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2020
Entry Details
US Patent

TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 286104BDBM286104(US9517228, Example 3 (2S,4′S) | US9987253, E...)
Affinity DataIC50: 100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2020
Entry Details
US Patent

TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 286106BDBM286106(US9517228, Example 4 (2S,4′S) | US9987253, E...)
Affinity DataIC50: 100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2020
Entry Details
US Patent

TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 286105BDBM286105(US9517228, Example 3a (2S,4′R) | US9987253, ...)
Affinity DataIC50: 750nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2020
Entry Details
US Patent

TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 286101BDBM286101(US9517228, Example 1a (4'R) | US9987253, Example 1...)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2020
Entry Details
US Patent

TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 286103BDBM286103(US9517228, Example 2a | US9987253, Example 2a | US...)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2020
Entry Details
US Patent

TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandChemical structure of BindingDB Monomer ID 286107BDBM286107(US9517228, Example 4a (2S,4′R) | US9987253, ...)
Affinity DataIC50: 1.00E+3nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2020
Entry Details
US Patent