Compile Data Set for Download or QSAR
Report error Found 91 Enz. Inhib. hit(s) with all data for entry = 9199
TargetRho-associated protein kinase 1(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322158BDBM322158(US10183931, Example 48 | 2-(3-(4-((1H-indazol-5-yl...)
Affinity DataKi:  10nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322176BDBM322176(US10183931, Example 176 | US10696660, Example 176 ...)
Affinity DataIC50: 13nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322158BDBM322158(US10183931, Example 48 | 2-(3-(4-((1H-indazol-5-yl...)
Affinity DataKi:  20nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322152BDBM322152(US10183931, Example 12 | (R)-2-(3-(4-((1H-indazol-...)
Affinity DataKi:  20nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322165BDBM322165(US10183931, Example 166 | US10696660, Example 166 ...)
Affinity DataIC50: 20nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322153BDBM322153(US10183931, Example 26 | 2-(3-(4-((1H-indazol-5-yl...)
Affinity DataKi:  30nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322153BDBM322153(US10183931, Example 26 | 2-(3-(4-((1H-indazol-5-yl...)
Affinity DataIC50: 30nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322167BDBM322167(US10183931, Example 168 | US10696660, Example 168 ...)
Affinity DataIC50: 30nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322174BDBM322174(US10183931, Example 17 | N-(3-(4-((1H-indazol-5-yl...)
Affinity DataIC50: 30nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322172BDBM322172(US10183931, Example 173 | US10696660, Example 173 ...)
Affinity DataIC50: 30nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322162BDBM322162(US10183931, Example 118 | 2-(3-(4-((1H-indazol-5-y...)
Affinity DataIC50: 40nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 448554BDBM448554(US10696660, Y-27263 | US11311541, Example Y-27263)
Affinity DataKi:  40nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322182BDBM322182(US10183931, Example 154 | N-(2-(3-(2-(isopropylami...)
Affinity DataIC50: 40nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322155BDBM322155(US11311541, Example SLx-2119 | US10696660, SLx-211...)
Affinity DataKi:  40nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322164BDBM322164(US10183931, Example 165 | US10696660, Example 165 ...)
Affinity DataIC50: 50nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322163BDBM322163(US10183931, Example 164 | US10696660, Example 164 ...)
Affinity DataIC50: 60nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 448554BDBM448554(US10696660, Y-27263 | US11311541, Example Y-27263)
Affinity DataKi:  60nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322166BDBM322166(US10183931, Example 167 | US10696660, Example 167 ...)
Affinity DataIC50: 60nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322169BDBM322169(US10183931, Example 170 | US10696660, Example 170 ...)
Affinity DataIC50: 70nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322152BDBM322152(US10183931, Example 12 | (R)-2-(3-(4-((1H-indazol-...)
Affinity DataKi:  70nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322160BDBM322160(US10183931, Example 5 | 2-(3-(4-((1H-indazol-5-yl)...)
Affinity DataIC50: 70nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322154BDBM322154(US10183931, Example 28 | 2-(3-(4-((1H-indazol-5-yl...)
Affinity DataIC50: 70nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322154BDBM322154(US10183931, Example 28 | 2-(3-(4-((1H-indazol-5-yl...)
Affinity DataKi:  80nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322170BDBM322170(US10183931, Example 171 | US10696660, Example 171 ...)
Affinity DataIC50: 80nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322161BDBM322161(US10183931, Example 163 | US10696660, Example 163 ...)
Affinity DataIC50: 80nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322184BDBM322184(US10183931, Example 159 | N-(2-(3-methoxyphenyl)-6...)
Affinity DataIC50: 100nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322171BDBM322171(US10183931, Example 172 | US10696660, Example 172 ...)
Affinity DataIC50: 120nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322157BDBM322157(US10183931, Example 14 | 2-(3-(4-((1H-indazol-5-yl...)
Affinity DataKi:  170nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322159BDBM322159(US10183931, Example 13 | (R)-2-(3-(4-((1H-indazol-...)
Affinity DataKi:  180nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322173BDBM322173(US10183931, Example 174 | US10696660, Example 174 ...)
Affinity DataIC50: 191nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322184BDBM322184(US10183931, Example 159 | N-(2-(3-methoxyphenyl)-6...)
Affinity DataIC50: 200nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322154BDBM322154(US10183931, Example 28 | 2-(3-(4-((1H-indazol-5-yl...)
Affinity DataKi:  260nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322158BDBM322158(US10183931, Example 48 | 2-(3-(4-((1H-indazol-5-yl...)
Affinity DataIC50: 300nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322181BDBM322181(US10183931, Example 179 | US10696660, Example 179 ...)
Affinity DataIC50: 310nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322158BDBM322158(US10183931, Example 48 | 2-(3-(4-((1H-indazol-5-yl...)
Affinity DataIC50: 330nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322183BDBM322183(US10183931, Example 22 | 3-(4-((1H-indazol-5-yl)am...)
Affinity DataIC50: 340nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322185BDBM322185(US10183931, Example 180 | US10696660, Example 180 ...)
Affinity DataIC50: 380nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322187BDBM322187(US10183931, Example 20 | 3-(4-((1H-indazol-5-yl)am...)
Affinity DataIC50: 400nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322158BDBM322158(US10183931, Example 48 | 2-(3-(4-((1H-indazol-5-yl...)
Affinity DataIC50: 470nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322175BDBM322175(US10183931, Example 175 | US10696660, Example 175 ...)
Affinity DataIC50: 500nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322155BDBM322155(US11311541, Example SLx-2119 | US10696660, SLx-211...)
Affinity DataKi:  500nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322152BDBM322152(US10183931, Example 12 | (R)-2-(3-(4-((1H-indazol-...)
Affinity DataIC50: 540nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322179BDBM322179(US10183931, Example 178 | US10696660, Example 178 ...)
Affinity DataIC50: 700nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322153BDBM322153(US10183931, Example 26 | 2-(3-(4-((1H-indazol-5-yl...)
Affinity DataIC50: 720nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322159BDBM322159(US10183931, Example 13 | (R)-2-(3-(4-((1H-indazol-...)
Affinity DataKi:  870nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322180BDBM322180(US10183931, Example 150 | N-(2-(4-(1-aminoethyl)ph...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322186BDBM322186(US10183931, Example 161 | N-(6-(2-(dimethylamino)e...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322158BDBM322158(US10183931, Example 48 | 2-(3-(4-((1H-indazol-5-yl...)
Affinity DataIC50: 1.00E+3nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 2(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 322155BDBM322155(US11311541, Example SLx-2119 | US10696660, SLx-211...)
Affinity DataIC50: 1.02E+3nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

TargetRho-associated protein kinase 1(Human)
Kadmon

US Patent
LigandChemical structure of BindingDB Monomer ID 448554BDBM448554(US10696660, Y-27263 | US11311541, Example Y-27263)
Affinity DataIC50: 1.13E+3nMAssay Description:Purified active ROCK1 and ROCK2 were obtained from Invitrogen (catalog numbers ROCK1, PV3691 and ROCK2, PV3759). The kit components include a coumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2021
Entry Details
US Patent

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