Compile Data Set for Download or QSAR
Report error Found 140 Enz. Inhib. hit(s) with all data for entry = 9330
LigandChemical structure of BindingDB Monomer ID 458418BDBM458418(US10744128, Compound 8)
Affinity DataEC50:  1nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458459BDBM458459(US10744128, Compound 45)
Affinity DataEC50:  1nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458458BDBM458458(US10744128, Compound 44)
Affinity DataEC50:  1nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458438BDBM458438(US10744128, Compound 24)
Affinity DataEC50:  2nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458411BDBM458411(US10744128, Compound 5 | US10744128, Compound 4)
Affinity DataEC50:  2nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458411BDBM458411(US10744128, Compound 5 | US10744128, Compound 4)
Affinity DataEC50:  2nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458463BDBM458463(US10744128, Compound 49)
Affinity DataEC50:  2nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458408BDBM458408(US10744128, Compound 3 | US10744128, Compound 2)
Affinity DataEC50:  2nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458477BDBM458477(US10744128, Compound 63)
Affinity DataEC50:  2nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458476BDBM458476(US10744128, Compound 62)
Affinity DataEC50:  2nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458456BDBM458456(US10744128, Compound 43 | US10744128, Compound 42)
Affinity DataEC50:  2nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458455BDBM458455(US10744128, Compound 41)
Affinity DataEC50:  2nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458419BDBM458419(US10744128, Compound 9)
Affinity DataEC50:  2nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458417BDBM458417(US10744128, Compound 7)
Affinity DataEC50:  3nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458415BDBM458415(US10744128, Compound 6)
Affinity DataEC50:  3nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458408BDBM458408(US10744128, Compound 3 | US10744128, Compound 2)
Affinity DataEC50:  3nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458445BDBM458445(US10744128, Compound 31)
Affinity DataEC50:  3nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458461BDBM458461(US10744128, Compound 47)
Affinity DataEC50:  3nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458446BDBM458446(US10744128, Compound 32)
Affinity DataEC50:  3nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458443BDBM458443(US10744128, Compound 29)
Affinity DataEC50:  3nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458444BDBM458444(US10744128, Compound 30)
Affinity DataEC50:  3nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458440BDBM458440(US10744128, Compound 26)
Affinity DataEC50:  3nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458420BDBM458420(US10744128, Compound 10)
Affinity DataEC50:  3nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458454BDBM458454(US10744128, Compound 40)
Affinity DataEC50:  4nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458465BDBM458465(US10744128, Compound 51)
Affinity DataEC50:  4nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458480BDBM458480(US10744128, Compound 66)
Affinity DataEC50:  4nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458478BDBM458478(US10744128, Compound 64)
Affinity DataEC50:  4nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458473BDBM458473(US10744128, Compound 59)
Affinity DataEC50:  4nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458474BDBM458474(US10744128, Compound 60)
Affinity DataEC50:  4nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458470BDBM458470(US10744128, Compound 56)
Affinity DataEC50:  5nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458475BDBM458475(US10744128, Compound 61)
Affinity DataEC50:  5nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458427BDBM458427(US10744128, Compound 13)
Affinity DataEC50:  5nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458460BDBM458460(US10744128, Compound 46)
Affinity DataEC50:  5nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458479BDBM458479(US10744128, Compound 65)
Affinity DataEC50:  6nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458448BDBM458448(US10744128, Compound 34)
Affinity DataEC50:  6nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458428BDBM458428(US10744128, Compound 14)
Affinity DataEC50:  6nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458471BDBM458471(US10744128, Compound 57)
Affinity DataEC50:  6nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458469BDBM458469(US10744128, Compound 55)
Affinity DataEC50:  7nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458447BDBM458447(US10744128, Compound 33)
Affinity DataEC50:  7nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458424BDBM458424(US10744128, Compound 11)
Affinity DataEC50:  7nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458429BDBM458429(US10744128, Compound 15)
Affinity DataEC50:  8nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458484BDBM458484(US10744128, Compound 70)
Affinity DataEC50:  9nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Samumed

US Patent
LigandChemical structure of BindingDB Monomer ID 458478BDBM458478(US10744128, Compound 64)
Affinity DataEC50:  9nMAssay Description:Briefly, recombinant GSK3β kinase, ATP and Ser/Thr peptide 09 are prepared in 1× Kinase buffer to final concentrations of 0.04 μg/mL, 46 &#...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458466BDBM458466(US10744128, Compound 52)
Affinity DataEC50:  9nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458425BDBM458425(US10744128, Compound 12)
Affinity DataEC50:  9nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458472BDBM458472(US10744128, Compound 58)
Affinity DataEC50:  9nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458449BDBM458449(US10744128, Compound 35)
Affinity DataEC50:  10nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458430BDBM458430(US10744128, Compound 19 | US10744128, Compound 16)
Affinity DataEC50:  12nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458467BDBM458467(US10744128, Compound 53)
Affinity DataEC50:  14nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 458441BDBM458441(US10744128, Compound 27)
Affinity DataEC50:  14nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Divis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

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