Compile Data Set for Download or QSAR
Report error Found 334 Enz. Inhib. hit(s) with all data for entry = 9336
TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418473BDBM418473(8-(1,3-Dimethyl-1H-pyrazol- 4-yl)-1-(3-fluoro-5-me...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418438BDBM418438(1-[5-(dimethylphosphinoylmethoxy)-3-fluoropyridin-...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418459BDBM418459(1-(3-Fluoro-5-methylpyridin- 2-yl)-7-methoxy-3-met...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418472BDBM418472(8-(1-Ethyl-1H-pyrazol-4-yl)- 1-(3-fluoro-5-methylp...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418448BDBM418448(8-(1,3-Dimethyl-1H-pyrazol- 4-yl)-1-(3-fluoropyrid...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418437BDBM418437(US10457677, Example 5 | US10745399, Example 5 | US...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418458BDBM418458(1-(3,5-Difluoropyridin-4-yl)- 8-(1-ethyl-1H-pyrazo...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418447BDBM418447(1-(3-Fluoro-5- methoxypyridin-4-yl)-7- methoxy-3-m...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418436BDBM418436(US10457677, Example 4 | US10745399, Example 4 | US...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418441BDBM418441(US10457677, Example 9 | US10745399, Example 9 | US...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418440BDBM418440(US10457677, Example 8 | US10745399, Example 8 | US...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418450BDBM418450(1-(3-Fluoro-5-methylpyridin- 4-yl)-7-methoxy-3-met...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418439BDBM418439(US10457677, Example 7 | US10745399, Example 7 | US...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418454BDBM418454(1-(3,5-Difluoropyridin-4-yl)- 7-methoxy-3-methyl-8...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418465BDBM418465(8-(1-Ethyl-1H-pyrazol-4-yl)- 1-(3-fluoropyridin-4-...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418443BDBM418443(US10457677, Example 11 | US10745399, Example 11 | ...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418453BDBM418453(1-(1,3-Dimethyl-1H-pyrazol- 4-yl)-8-(1-ethyl-1H-py...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418442BDBM418442(US10457677, Example 10 | US10745399, Example 10 | ...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418477BDBM418477(7-Methoxy-3-methyl-1-(3- methyl-1H-pyrazol-4-yl)-8...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418452BDBM418452(1-(3-Fluoro-5-methylpyridin- 2-yl)-7-methoxy-3-met...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418470BDBM418470(1-(5-Fluoropyrimidin-2-yl)-7- methoxy-3-methyl-8-(...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418446BDBM418446(US10457677, Example 14 | US10745399, Example 14 | ...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418457BDBM418457(1-(3-Ethyl-5-fluoropyridin-4- yl)-8-(1-ethyl-1H-py...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418435BDBM418435(1-[5-(azetidin-3-ylmethoxy)-3-fluoropyridin-2-yl]-...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418445BDBM418445(US10457677, Example 13 | US10745399, Example 13 | ...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418456BDBM418456(8-(1-Ethyl-1H-pyrazol-4-yl)- 1-(3-fluoropyridin-2-...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418434BDBM418434(US10457677, Example 2 | US10745399, Example 2 | US...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418444BDBM418444(US10457677, Example 12 | US10745399, Example 12 | ...)
Affinity DataIC50: 1nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418460BDBM418460(7-Methoxy-1-(3-methoxy- pyridin-4-yl)-3-methyl-8-(...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418449BDBM418449(7-Methoxy-3-methyl-1-(1- methyl-1H-pyrazol-4-yl)-8...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418489BDBM418489(7-Methoxy-3-methyl-8-(1- methyl-1H-pyrazol-4-yl)-1...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418487BDBM418487(1-(3-Fluoropyridin-2-yl)-7- methoxy-3-methyl-8-(1-...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418471BDBM418471(7-Methoxy-3-methyl-8-(1H- pyrazol-4-yl)-1-[1- (tet...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418462BDBM418462(7-Methoxy-3-methyl-1-(2- methylthiazol-4-yl)-8-(1H...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418475BDBM418475(7-Methoxy-3-methyl-1-(2- methyl-2H-pyrazol-3-yl)-8...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418451BDBM418451(7-Methoxy-3-methyl-1-(3- methylpyridin-4-yl)-8-(1H...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418461BDBM418461(1-(3-Fluoropyridin-2-yl)-7- methoxy-3-methyl-8-(5-...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418474BDBM418474(7-Methoxy-3-methyl-8-(1- methyl-1H-pyrazol-4-yl)-1...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418491BDBM418491(7-Methoxy-3-methyl-8-(1- methyl-1H-pyrazol-4-yl)-1...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418490BDBM418490(1-(3-Ethyl-5-methylpyridin- 4-yl)-7-methoxy-3-meth...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418433BDBM418433(US10457677, Example 1 | US10745399, Example 1 | US...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418496BDBM418496(1-(3-Chloropyridin-4-yl)-7- methoxy-3-methyl-8-(1-...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418464BDBM418464(7-Methoxy-1-(3-methoxy- pyridin-4-yl)-3-methyl-8- ...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418480BDBM418480(5-Fluoro-4-[7-methoxy-3- methyl-8-(1-methyl-1H- py...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418495BDBM418495(7-Methoxy-3-methyl-1-(1- methyl-1H-imidazol-4-yl)-...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418463BDBM418463(1-(5-Fluoropyrimidin-4-yl)-7- methoxy-3-methyl-8-(...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418494BDBM418494(7-Methoxy-3-methyl-8-(1- methyl-1H-pyrazol-4-yl)-1...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418485BDBM418485(7-Methoxy-3-methyl-1-(2- methyl-2H-pyrazol-3-yl)-8...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418483BDBM418483(7-Methoxy-3-methyl-8-(1- methyl-1H-pyrazol-4-yl)-1...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

TargetSerine-protein kinase ATM(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 418469BDBM418469(1-(3-Fluoropyridin-4-yl)-7- methoxy-3-methyl-8-(1-...)
Affinity DataIC50: 10nMAssay Description:The IC50 value was determined with the aid of a biochemical ATM kinase assay. The assay consists of two steps: the enzymatic reaction and the detecti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2021
Entry Details
US Patent

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