Compile Data Set for Download or QSAR
Report error Found 98 Enz. Inhib. hit(s) with all data for entry = 9517
LigandChemical structure of BindingDB Monomer ID 426381BDBM426381(US10526325, Compound A57 | US10829489, Compound A5...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426378BDBM426378(US10526325, Compound A54 | US10829489, Compound A5...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426378BDBM426378(US10526325, Compound A54 | US10829489, Compound A5...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426376BDBM426376(US10526325, Compound A52 | US10829489, Compound A5...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426328BDBM426328(US10526325, Compound A5 | US10829489, Compound A5 ...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426328BDBM426328(US10526325, Compound A5 | US10829489, Compound A5 ...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426327BDBM426327(US10526325, Compound A4 | US10829489, Compound A4 ...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426327BDBM426327(US10526325, Compound A4 | US10829489, Compound A4 ...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426326BDBM426326(US10526325, Compound A3 | US10829489, Compound A3 ...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426326BDBM426326(US10526325, Compound A3 | US10829489, Compound A3 ...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426324BDBM426324(US10526325, Compound A1 | US10829489, Compound A1 ...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426324BDBM426324(US10526325, Compound A1 | US10829489, Compound A1 ...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 472696BDBM472696((2R)-3,3,3-trifluoro-1-[1-(4-fluorophenyl)-7-methy...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 472696BDBM472696((2R)-3,3,3-trifluoro-1-[1-(4-fluorophenyl)-7-methy...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426333BDBM426333(US10526325, Compound A10 | US10829489, Compound A1...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426333BDBM426333(US10526325, Compound A10 | US10829489, Compound A1...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426332BDBM426332(US10526325, Compound A9 | (2R)-1-[1-(4-chloropheny...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426332BDBM426332(US10526325, Compound A9 | (2R)-1-[1-(4-chloropheny...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426330BDBM426330(US10526325, Compound A7 | US10829489, Compound A7 ...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426330BDBM426330(US10526325, Compound A7 | US10829489, Compound A7 ...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426329BDBM426329(US10526325, Compound A6 | US10829489, Compound A6 ...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426346BDBM426346(US10526325, Compound A22 | US10829489, Compound A2...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426346BDBM426346(US10526325, Compound A22 | US10829489, Compound A2...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426344BDBM426344(US10526325, Compound A20 | US10829489, Compound A2...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426344BDBM426344(US10526325, Compound A20 | US10829489, Compound A2...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426342BDBM426342(US10526325, Compound A18 | US10829489, Compound A1...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426342BDBM426342(US10526325, Compound A18 | US10829489, Compound A1...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 472700BDBM472700((R)-3,3,3-Trifluoro-2-hydroxy-2-methyl-1-(7-methyl...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 472700BDBM472700((R)-3,3,3-Trifluoro-2-hydroxy-2-methyl-1-(7-methyl...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426338BDBM426338(US10526325, Compound A14 | US10829489, Compound A1...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426338BDBM426338(US10526325, Compound A14 | US10829489, Compound A1...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426358BDBM426358(US10526325, Compound A34 | US10829489, Compound A3...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426356BDBM426356(US10526325, Compound A32 | US10829489, Compound A3...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426356BDBM426356(US10526325, Compound A32 | US10829489, Compound A3...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426354BDBM426354(US10526325, Compound A30 | US10829489, Compound A3...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426354BDBM426354(US10526325, Compound A30 | US10829489, Compound A3...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426352BDBM426352(US10526325, Compound A28 | US10829489, Compound A2...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426348BDBM426348(US10526325, Compound A24 | US10829489, Compound A2...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426348BDBM426348(US10526325, Compound A24 | US10829489, Compound A2...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 472850BDBM472850((R)-3,3,3-Trifluoro-2-hydroxy-2-methyl-1-(3-phenyl...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426366BDBM426366(US10526325, Compound A42 | US10829489, Compound A4...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426364BDBM426364(US10526325, Compound A40 | US10829489, Compound A4...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426364BDBM426364(US10526325, Compound A40 | US10829489, Compound A4...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426362BDBM426362(US10526325, Compound A38 | US10829489, Compound A3...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426362BDBM426362(US10526325, Compound A38 | US10829489, Compound A3...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426358BDBM426358(US10526325, Compound A34 | US10829489, Compound A3...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426375BDBM426375(US10526325, Compound A51 | US10829489, Compound A5...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426376BDBM426376(US10526325, Compound A52 | US10829489, Compound A5...)
Affinity DataIC50: 300nMAssay Description:The PDC inactivation assay is performed in Greiner 384-well microtiter plates and is used for high throughput screen. 4 μl of PDHK2 (human, rec,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426374BDBM426374(US10526325, Compound A50 | US10829489, Compound A5...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 426373BDBM426373(US10526325, Compound A49 | US10829489, Compound A4...)
Affinity DataKd: <300nMAssay Description:ITC measurements were performed with a VP-ITC micro calorimeter (Microcal, LLC/GE Healthcare Bio-Sciences AB, Uppsala, Sweden). In general titrations...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
US Patent

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