Compile Data Set for Download or QSAR
Report error Found 106 Enz. Inhib. hit(s) with all data for entry = 9562
TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474403BDBM474403(US10858373, Example 1 | 1,1,1,3,3,3-Hexafluoroprop...)
Affinity DataIC50: 0.259nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474408BDBM474408(US10858373, Example 6 | 1,1,1,3,3,3-Hexafluoroprop...)
Affinity DataIC50: 0.470nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474444BDBM474444(US10858373, Example 42)
Affinity DataIC50: 0.587nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474454BDBM474454(US10858373, Example 52)
Affinity DataIC50: 0.666nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474429BDBM474429(US10858373, Example 27)
Affinity DataIC50: 0.679nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474416BDBM474416(US10858373, Example 14 | 1,1,1,3,3,3-Hexafluoropro...)
Affinity DataIC50: 0.942nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474404BDBM474404(US10858373, Example 2 | 1,1,1,3,3,3-Hexafluoroprop...)
Affinity DataIC50: 1nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474434BDBM474434(US10858373, Example 32)
Affinity DataIC50: 1.08nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474435BDBM474435(US10858373, Example 33)
Affinity DataIC50: 1.21nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474443BDBM474443(US10858373, Example 41)
Affinity DataIC50: 1.25nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474442BDBM474442(US10858373, Example 40)
Affinity DataIC50: 1.43nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474451BDBM474451(US10858373, Example 49)
Affinity DataIC50: 1.45nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474440BDBM474440(US10858373, Example 38)
Affinity DataIC50: 2.19nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474430BDBM474430(US10858373, Example 28)
Affinity DataIC50: 2.22nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474433BDBM474433(US10858373, Example 31)
Affinity DataIC50: 2.26nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474413BDBM474413(US10858373, Example 11 | 1,1,1,3,3,3-Hexafluoropro...)
Affinity DataIC50: 2.46nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474452BDBM474452(US10858373, Example 50)
Affinity DataIC50: 2.46nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474438BDBM474438(US10858373, Example 36)
Affinity DataIC50: 2.79nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474439BDBM474439(US10858373, Example 37)
Affinity DataIC50: 3.03nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474403BDBM474403(US10858373, Example 1 | 1,1,1,3,3,3-Hexafluoroprop...)
Affinity DataIC50: 3.09nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474410BDBM474410(US10858373, Example 8 | 1,1,1,3,3,3-Hexafluoroprop...)
Affinity DataIC50: 3.29nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474416BDBM474416(US10858373, Example 14 | 1,1,1,3,3,3-Hexafluoropro...)
Affinity DataIC50: 3.63nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474441BDBM474441(US10858373, Example 39)
Affinity DataIC50: 4.04nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474408BDBM474408(US10858373, Example 6 | 1,1,1,3,3,3-Hexafluoroprop...)
Affinity DataIC50: 4.39nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474414BDBM474414(US10858373, Example 12 | 1,1,1,3,3,3-Hexafluoropro...)
Affinity DataIC50: 4.90nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474444BDBM474444(US10858373, Example 42)
Affinity DataIC50: 4.93nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474429BDBM474429(US10858373, Example 27)
Affinity DataIC50: 6.25nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474417BDBM474417(US10858373, Example 15)
Affinity DataIC50: 7.86nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474404BDBM474404(US10858373, Example 2 | 1,1,1,3,3,3-Hexafluoroprop...)
Affinity DataIC50: 7.94nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474454BDBM474454(US10858373, Example 52)
Affinity DataIC50: 8.04nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474451BDBM474451(US10858373, Example 49)
Affinity DataIC50: 8.34nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474405BDBM474405(US10858373, Example 3 | 1,1,1,3,3,3-Hexafluoroprop...)
Affinity DataIC50: 8.49nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474455BDBM474455(US10858373, Example 53)
Affinity DataIC50: 10.1nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474430BDBM474430(US10858373, Example 28)
Affinity DataIC50: 10.3nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474418BDBM474418(US10858373, Example 16)
Affinity DataIC50: 10.4nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474419BDBM474419(US10858373, Example 17)
Affinity DataIC50: 10.5nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474443BDBM474443(US10858373, Example 41)
Affinity DataIC50: 12nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474434BDBM474434(US10858373, Example 32)
Affinity DataIC50: 13.7nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474420BDBM474420(US10858373, Example 18)
Affinity DataIC50: 14nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474435BDBM474435(US10858373, Example 33)
Affinity DataIC50: 15nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474409BDBM474409(US10858373, Example 7 | N-[(3R)-8-{[(2,5-Dioxopyrr...)
Affinity DataIC50: 15.6nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474413BDBM474413(US10858373, Example 11 | 1,1,1,3,3,3-Hexafluoropro...)
Affinity DataIC50: 17.6nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474452BDBM474452(US10858373, Example 50)
Affinity DataIC50: 19nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474406BDBM474406(US10858373, Example 4)
Affinity DataIC50: 20.3nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474433BDBM474433(US10858373, Example 31)
Affinity DataIC50: 20.8nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474440BDBM474440(US10858373, Example 38)
Affinity DataIC50: 22nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474442BDBM474442(US10858373, Example 40)
Affinity DataIC50: 22.9nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474449BDBM474449(US10858373, Example 47)
Affinity DataIC50: 23nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474439BDBM474439(US10858373, Example 37)
Affinity DataIC50: 25.8nMAssay Description:Assessment of MAGL inhibition utilizes human recombinant Monoacylglycerol Lipase and the fluorogenic substrate 7-hydroxycoumarinyl arachidonate (7-HC...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

TargetMonoglyceride lipase(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 474421BDBM474421(US10858373, Example 19)
Affinity DataIC50: 28.5nMAssay Description:T = 30 minutes.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2021
Entry Details
US Patent

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