Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 9613
LigandChemical structure of BindingDB Monomer ID 476730BDBM476730(US10870651, Compound 118)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476729BDBM476729(US10870651, Compound 117)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476728BDBM476728(US10870651, Compound 116)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476727BDBM476727(US10870651, Compound 115)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476726BDBM476726(US10870651, Compound 114)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476725BDBM476725(US10870651, Compound 113)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476724BDBM476724(US10870651, Compound 112)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476722BDBM476722(US10870651, Compound 110)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476721BDBM476721(US10870651, Compound 109)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476720BDBM476720(US10870651, Compound 108)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476719BDBM476719(US10870651, Compound 107)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476718BDBM476718(US10870651, Compound 105)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476717BDBM476717(US10870651, Compound 104)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476716BDBM476716(US10870651, Compound 103)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476742BDBM476742(US10870651, Compound 234)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476741BDBM476741(US10870651, Compound 233)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476740BDBM476740(US10870651, Compound 232)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476739BDBM476739(US10870651, Compound 231)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476738BDBM476738(US10870651, Compound 222)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476737BDBM476737(US10870651, Compound 217)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476736BDBM476736(US10870651, Compound 216)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476735BDBM476735(US10870651, Compound 215)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent
PDB3D3D Structure (crystal)
LigandChemical structure of BindingDB Monomer ID 476734BDBM476734(US10870651, Compound 214)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476733BDBM476733(US10870651, Compound 123)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476732BDBM476732(US10870651, Compound 120)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476731BDBM476731(US10870651, Compound 119)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476750BDBM476750(US10870651, Compound 241)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50526807BDBM50526807(CHEMBL4467048 | US10870651, Compound 102)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50526803BDBM50526803(CHEMBL4434871 | US10870651, Compound 101)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
Dana-Farber Cancer Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 50526803BDBM50526803(CHEMBL4434871 | US10870651, Compound 101)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Dana-Farber Cancer Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 50526803BDBM50526803(CHEMBL4434871 | US10870651, Compound 101)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

TargetProtein kinase C theta type(Human)
Dana-Farber Cancer Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 50526803BDBM50526803(CHEMBL4434871 | US10870651, Compound 101)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

TargetTyrosine-protein kinase Fgr(Human)
Dana-Farber Cancer Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 50526803BDBM50526803(CHEMBL4434871 | US10870651, Compound 101)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

TargetSerine/threonine-protein kinase Chk2(Human)
Dana-Farber Cancer Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 50526803BDBM50526803(CHEMBL4434871 | US10870651, Compound 101)
Affinity DataIC50: 100nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476744BDBM476744(US10870651, Compound 236)
Affinity DataIC50: 300nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476723BDBM476723(US10870651, Compound 111)
Affinity DataIC50: 300nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476756BDBM476756(US10870651, Compound 246)
Affinity DataIC50: 300nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476714BDBM476714(US10870651, Compound 106)
Affinity DataIC50: 300nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476745BDBM476745(US10870651, Compound 238 | US10870651, Compound 23...)
Affinity DataIC50: 500nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476745BDBM476745(US10870651, Compound 238 | US10870651, Compound 23...)
Affinity DataIC50: 500nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476743BDBM476743(US10870651, Compound 235)
Affinity DataIC50: 500nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476755BDBM476755(US10870651, Compound 245)
Affinity DataIC50: 500nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476754BDBM476754(US10870651, Compound 244)
Affinity DataIC50: 500nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476753BDBM476753(US10870651, Compound 243)
Affinity DataIC50: 500nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476752BDBM476752(US10870651, Compound 242)
Affinity DataIC50: 500nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476747BDBM476747(US10870651, Compound 240 | US10870651, Compound 23...)
Affinity DataIC50: 500nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 476747BDBM476747(US10870651, Compound 240 | US10870651, Compound 23...)
Affinity DataIC50: 500nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

TargetMaternal embryonic leucine zipper kinase(Human)
Dana-Farber Cancer Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 476714BDBM476714(US10870651, Compound 106)
Affinity DataIC50: 550nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

TargetMaternal embryonic leucine zipper kinase(Human)
Dana-Farber Cancer Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 50526803BDBM50526803(CHEMBL4434871 | US10870651, Compound 101)
Affinity DataIC50: 550nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

TargetHomeodomain-interacting protein kinase 4(Human)
Dana-Farber Cancer Institute

US Patent
LigandChemical structure of BindingDB Monomer ID 50526803BDBM50526803(CHEMBL4434871 | US10870651, Compound 101)
Affinity DataIC50: 550nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/26/2021
Entry Details
US Patent

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