Compile Data Set for Download or QSAR
Report error Found 91 Enz. Inhib. hit(s) with all data for entry = 9696
LigandChemical structure of BindingDB Monomer ID 482266BDBM482266(US10918645, Example 65)
Affinity DataIC50: 4nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482288BDBM482288(US10918645, Example 91 | 8-ethyl-4-(tetrahydro-2H-...)
Affinity DataIC50: 6nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482268BDBM482268(US10918645, Example 66 | US10918645, Example 67)
Affinity DataIC50: 7nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482275BDBM482275(US10918645, Example 71 | 1-methyl-9-(tetrahydro-2H...)
Affinity DataIC50: 11nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482286BDBM482286(US10918645, Example 90 | 8-methyl-4-(tetrahydro-2H...)
Affinity DataIC50: 12nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482290BDBM482290(US10918645, Example 92 | 8-isopropyl-4-(tetrahydro...)
Affinity DataIC50: 13nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482277BDBM482277(US10918645, Example 72 | 2-ethyl-9-(tetrahydro-2H-...)
Affinity DataIC50: 15nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482283BDBM482283(US10918645, Example 75 | 1-isopropyl-9-(tetrahydro...)
Affinity DataIC50: 16nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482244BDBM482244(US10918645, Example 51 | 4-cyclobutyl-5,11-dihydro...)
Affinity DataIC50: 20nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482279BDBM482279(US10918645, Example 73 | 1-ethyl-9-(tetrahydro-2H-...)
Affinity DataIC50: 21nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482274BDBM482274(US10918645, Example 83 | 9-(1-isopropylpiperidin-4...)
Affinity DataIC50: 23nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482273BDBM482273(US10918645, Example 70 | 2-methyl-9-(tetrahydro-2H...)
Affinity DataIC50: 23nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482268BDBM482268(US10918645, Example 66 | US10918645, Example 67)
Affinity DataIC50: 26nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482278BDBM482278(US10918645, Example 86 | 2-ethyl-9-(1-isopropylpip...)
Affinity DataIC50: 29nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482236BDBM482236(US10918645, Example 47 | US10918645, Example 33 | ...)
Affinity DataIC50: 30nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482282BDBM482282(US10918645, Example 88 | 2-isopropyl-9-(1-isopropy...)
Affinity DataIC50: 31nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482252BDBM482252(US10918645, Example 55 | US10918645, Example 42 | ...)
Affinity DataIC50: 31nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482248BDBM482248(US10918645, Example 53 | 4-phenyl-5,11-dihydro-4H-...)
Affinity DataIC50: 33nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482246BDBM482246(US10918645, Example 52 | 4-cyclopentyl-5,11-dihydr...)
Affinity DataIC50: 33nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482234BDBM482234(US10918645, Example 46 | 4-ethyl-5,11-dihydro- 4H-...)
Affinity DataIC50: 34nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482285BDBM482285(US10918645, Example 68)
Affinity DataIC50: 34nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482244BDBM482244(US10918645, Example 51 | 4-cyclobutyl-5,11-dihydro...)
Affinity DataIC50: 39nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482272BDBM482272(US10918645, Example 82 | 9-(1-isopropylpiperidin-4...)
Affinity DataIC50: 39nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482287BDBM482287(US10918645, Example 81 | 2-isopropyl-9-(1-methylpi...)
Affinity DataIC50: 40nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482238BDBM482238(US10918645, Example 48 | US10918645, Example 34 | ...)
Affinity DataIC50: 41nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482260BDBM482260(US10918645, Example 59 | 8-fluoro-4-(tetrahydro-2H...)
Affinity DataIC50: 46nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482289BDBM482289(US10918645, Example 84 | 1-isopropyl-9-(1-(2-metho...)
Affinity DataIC50: 46nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482262BDBM482262(US10918645, Example 60 | 4-(tetrahydro-2H-pyran-4-...)
Affinity DataIC50: 47nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482258BDBM482258(US10918645, Example 58 | US10918645, Example 44 | ...)
Affinity DataIC50: 48nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482234BDBM482234(US10918645, Example 46 | 4-ethyl-5,11-dihydro- 4H-...)
Affinity DataIC50: 49nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482284BDBM482284(US10918645, Example 89)
Affinity DataIC50: 49nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482281BDBM482281(US10918645, Example 74 | 2-isopropyl-9-(tetrahydro...)
Affinity DataIC50: 50nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482276BDBM482276(US10918645, Example 85 | 1-ethyl-9-(1-isopropylpip...)
Affinity DataIC50: 50nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482252BDBM482252(US10918645, Example 55 | US10918645, Example 42 | ...)
Affinity DataIC50: 50nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482236BDBM482236(US10918645, Example 47 | US10918645, Example 33 | ...)
Affinity DataIC50: 54nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482264BDBM482264(US10918645, Example 61 | 8-fluoro-4-(tetrahydro-2H...)
Affinity DataIC50: 57nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482254BDBM482254(US10918645, Example 56 | 4-(1-isopropylpiperidin- ...)
Affinity DataIC50: 58nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482280BDBM482280(US10918645, Example 87 | 1-isopropyl-9-(1-isopropy...)
Affinity DataIC50: 62nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482240BDBM482240(US10918645, Example 49 | 4-isobutyl-5,11-dihydro-4...)
Affinity DataIC50: 67nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482238BDBM482238(US10918645, Example 48 | US10918645, Example 34 | ...)
Affinity DataIC50: 68nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482232BDBM482232(US10918645, Example 45 | US10918645, Example 31)
Affinity DataIC50: 71nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482258BDBM482258(US10918645, Example 58 | US10918645, Example 44 | ...)
Affinity DataIC50: 74nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482240BDBM482240(US10918645, Example 49 | 4-isobutyl-5,11-dihydro-4...)
Affinity DataIC50: 75nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482245BDBM482245(US10918645, Example 26 | 6-(1-methylpiperidin- 4-y...)
Affinity DataIC50: 91nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482232BDBM482232(US10918645, Example 45 | US10918645, Example 31)
Affinity DataIC50: 110nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482242BDBM482242(US10918645, Example 50 | 4-(sec-butyl)-5,11-dihydr...)
Affinity DataIC50: 120nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482239BDBM482239(US10918645, Example 22 | 6-cyclobutyl-6,7,8,9- tet...)
Affinity DataIC50: 140nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482250BDBM482250(US10918645, Example 54 | 4-benzyl-5,11-dihydro-4H-...)
Affinity DataIC50: 140nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482249BDBM482249(US10918645, Example 29 | 6-(tetrahydro-2H-pyran- 4...)
Affinity DataIC50: 150nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 482241BDBM482241(US10918645, Example 23 | 6-cyclopentyl-6,7,8,9-tet...)
Affinity DataIC50: 150nMAssay Description:TTBK1 (5-20 mU diluted in 50 mM Tris pH 7.5, 0.1 mM EGTA, 0.1% β-mercaptoethanol, 1 mg/ml BSA, 10 mM DTT) is assayed against RRKDLHDDEEDEAMSITA ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/2/2021
Entry Details
US Patent

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